A copper‐catalyzed, intramolecular borylative cyclization of vinyl arenes with imines is
reported, which affords enantio‐enriched indolines as a single diastereomer under mild …

The development of an efficient, straightforward approach for access to a wide range of
enantioenriched boron-containing 2, 3-disubstituted indolines via highly chemo-, diastereo …

A copper (I)-catalyzed dearomative borylation of N-alkoxycarbonyl protected indole-3-
carboxylates has been developed. The boron addition in this reaction occurred …

Cu‐catalyzed intramolecular borylation‐cross coupling reaction of alkenes was developed.
Racemic and chiral borylated indolines were achieved by borylation‐cross coupling of …

Copper (I)-catalyzed enantioselective borylation of α, β-unsaturated N-acylindoles as well as
N-acylpyrroles was efficiently achieved by means of bis (pinacolato) diboron (B2pin2) …

The first Cu-catalyzed asymmetric borylative cyclization of cyclohexadienone-containing 1, 6-
enynes is achieved through a tandem process: selective β-borylation of propargylic ether …

The enantioselective borylative dearomatization of a heteroaromatic compound has been
achieved using a copper (I) catalyst and a diboron reagent. This reaction involves the regio …

We report a Cu (II)-(S, S)-i Pr-FOXAP-catalyzed borylative Michael/Michael addition cascade
cyclization of unsymmetrical dienone for the synthesis of highly substituted and …

Copper (I)-catalyzed diastereoselective borylative exo-cyclization of alkenyl ketones with bis
(pinacolato) diboron is reported. The reaction of alkenyl aryl ketones under a CuCl/Xantphos …

We report broadly applicable copper catalytic conditions for the diastereoselective and
enantioselective 1, 2-addition of 1, 1-diborylalkanes to cyclic ketimines and α-imino esters …