β-(2-aminophenyl)-α, β-ynones can quickly give functionalized 2, 4-disubstituted quinolines
through tandem nucleophic addition/annulations reactions. Acid-catalysed cyclization of β-(2 …

A two-stage “tandem strategy” for the regiocontrolled synthesis of very highly substituted
quinolines is described. Benzannulation based on the reaction of cyclobutenones or diazo …

A catalyst-free synthetic approach is described for the synthesis of 4-quinolone derivatives
through a tandem amination/conjugated Michael addition sequence of 1-(2-fluorophenyl) …

β-(2-Aminophenyl)-α, β-ynones react with enamines of cyclic ketones by domino [2+ 2]
cycloaddition/annelation reaction giving rise to bicyclo [4.2. 0]-octane [7, 8-c]-2-aryl …

Concise and efficient syntheses of various trans-2, 3-disubstituted-2, 3-dihydro-4-quinolones
have been achieved via tandem Hofmann-type rearrangement of 2-alkynylbenzamides …

Regioselective synthesis of 3-bromoquinoline derivatives was achieved via a formal [4+ 2]-
cycloaddition between N-aryliminium ion, generated from arylmethyl azides, and 1 …

A review of the recent literature is given focusing on synthetic approaches to 1, 2, 3, 4-
tetrahydroquinolines, 2, 3-dihydro-4 (1 H)-quinolinones and 4 (1 H)-quinolinones using …

The regioselective construction of functionalized quinolines by the three-component
reactions of enaminones, aldehydes and anilines is accomplished. Unlike conventional …

The 3, 4, 8-trisubstituted quinoline derivatives 2-butyryl-8-methoxy-4-[(2-methylphenyl)
amino] quinoline and 3-butyryl-8-(2-hydroxyethoxy)-4-[(2-methylphenyl) amino] quinoline …

A practical synthesis of 7-mono-substituted quinolines has been achieved. Selective
reduction of the inexpensive commercial reagent 4, 7-dichloroquinoline affords 7 …