An acid-promoted cyclization of α-azidobenzyl ketones has been developed for the
synthesis of 6-substituted quinoline derivatives. A variety of synthetically useful 6-OTf or …

A protocol involving intramolecular formal [4+ 2]‐cycloaddition of in situ generated o‐aza‐
quinone methide for the facile synthesis of 1, 4‐heterocycle‐fused quinoline motifs is …

A novel acid/base-co-catalyzed tandem cyclization of various ketones with o-amino-
benzylamines employing molecular oxygen as the clean oxidant has been described. The …

The intramolecular cyclization of allylamines and ketones was achieved in the presence of
potassium tert‐butoxide and N, N‐dimethylformamide. A series of 4‐arylquinolines was …

A two-stage “tandem strategy” for the regiocontrolled synthesis of very highly substituted
quinolines is described. Benzannulation based on the reaction of cyclobutenones or diazo …

A one-pot process to introduce diazoacetoacetate functionality into quinoline was identified
with excellent yield and regioselectivity. An intramolecular cyclopropanation of the resulting …

Regioselective synthesis of 3-bromoquinoline derivatives was achieved via a formal [4+ 2]-
cycloaddition between N-aryliminium ion, generated from arylmethyl azides, and 1 …

A practical Cu-catalyzed cascade cyclization of o-halobenzoate with enaminones to
construct isoquinolinone derivatives is described. The process involves a Cu-catalyzed …

Abstract Reductive cyclization of ω-(8-quinolyloxy) alkyl esters by zinc in acetic acid is
shown to constitute a convenient methodology for the synthesis of oxazino-or oxazepino …

A new and efficient strategy for the synthesis of substituted quinolines via electrophilic
cyclization is developed. The intramolecular cyclization of 1-azido-2-(2-propynyl) benzene 1 …