An efficient and rapid synthesis of multiply substituted quinolines is described. This method
is enabled by a three-component cascade annulation of readily available aryl diazonium …

Synthesis of 3‐Iodoquinolines by Copper‐Catalyzed Tandem Annulation from
Diaryliodoniums, Nitriles, and 1‐Iodoalkynes - Wang - 2016 - Advanced Synthesis & …

An efficient single-step approach toward the synthesis of 2-alkylquinolines is described.
Through a Lewis acid mediated [3+ 3] annulation reaction between 3-ethoxycyclobutanones …

One-pot synthesis of 3-aryl-4 (3H)-quinazolinones has been realized through a cascade
annulation. Reaction of aryldiazonium salt with a nitrile provides in situ generation of a …

A convergent, catalytic asymmetric formal [4+ 2] annulation for the synthesis of
dihydroquinolones has been developed. Carboxylic acids can be employed as precursors to …

A copper (I)-catalyzed protocol is developed for the synthesis of various 2, 3-
diaroylquinolines starting from achiral ammonium salts and anthranils through [4+ 1+ 1] …

A two-stage “tandem strategy” for the regiocontrolled synthesis of very highly substituted
quinolines is described. Benzannulation based on the reaction of cyclobutenones or diazo …

An oxidative annulation for the synthesis of 2, 4-diarylquinolines from o-allylanilines is
disclosed that uses recyclable reagent Chloranil as the oxidant. The corresponding products …

An efficient one-pot approach to multiple substituted quinazolines with diaryliodonium salt 1,
and two nitriles 2 has been presented. The reaction enables great flexibility of the …

A transition metal-free protocol has been developed for the synthesis of 3-acyl quinolines
through aza-Michael addition and intramolecular annulation of enaminones with anthranils …