Primary structure and function of an A kinase anchoring protein associated with calcium channels

PC Gray, BD Johnson, RE Westenbroek, LG Hays… - Neuron, 1998 - cell.com
PC Gray, BD Johnson, RE Westenbroek, LG Hays, JR Yates, T Scheuer, WA Catterall…
Neuron, 1998cell.com
Rapid, voltage-dependent potentiation of skeletal muscle L-type calcium channels requires
phosphorylation by cAMP-dependent protein kinase (PKA) anchored via an A kinase
anchoring protein (AKAP). Here we report the isolation, primary sequence determination,
and functional characterization of AKAP15, a lipid-anchored protein of 81 amino acid
residues with a single amphipathic helix that binds PKA. AKAP15 colocalizes with L-type
calcium channels in transverse tubules and is associated with L-type calcium channels in …
Abstract
Rapid, voltage-dependent potentiation of skeletal muscle L-type calcium channels requires phosphorylation by cAMP-dependent protein kinase (PKA) anchored via an A kinase anchoring protein (AKAP). Here we report the isolation, primary sequence determination, and functional characterization of AKAP15, a lipid-anchored protein of 81 amino acid residues with a single amphipathic helix that binds PKA. AKAP15 colocalizes with L-type calcium channels in transverse tubules and is associated with L-type calcium channels in transfected cells. A peptide fragment of AKAP15 encompassing the RII-binding domain blocks voltage-dependent potentiation. These results indicate that AKAP15 targets PKA to the calcium channel and plays a critical role in voltage-dependent potentiation and regulation of skeletal muscle contraction. The expression of AKAP15 in the brain and heart suggests that it may mediate rapid PKA regulation of L-type calcium channels in neurons and cardiac myocytes.
cell.com
以上显示的是最相近的搜索结果。 查看全部搜索结果