Synthesis of Substituted 1H-Indazoles by Pyrazole Annelation to an Arene

AK Garkushenko, OP Sorokina, GA Kryuchkova… - Chemistry of …, 2013 - Springer
Substituted 1 H-indazoles have been synthesized by reductive intramolecular
heterocyclization of 2, 4-di-aroyl-N-nitrosomethylanilines and 2, 4-diacetyl-N …

Synthesis of 3-R2-4-R1-acetyl-(ethoxycarbonyl)-6-hydroxy-6-methylindazoles

VV Sorokin, AV Grigor'ev, AK Ramazanov… - Chemistry of …, 1999 - Springer
It was discovered that functionally substituted tetrahydroindazoles can be aromatized by the
action of sulfur. Previously unknown 3-R 2-4-R 1-5-acetyl (ethoxycarbonyl)-6 …

N,N-Bond-Forming Heterocyclization:  Synthesis of 3-Alkoxy-2H-indazoles

AD Mills, MZ Nazer, MJ Haddadin… - The Journal of organic …, 2006 - ACS Publications
A one-step heterocyclization of o-nitrobenzylamines to 3-alkoxy-2 H-indazoles is reported.
The electronic nature of the nitrophenyl group, the steric and electronic nature of the R1 …

Simple Synthesis of 3-Alkyl-1H-Indazoles Having Functional Groups At the ω-Position

K Sasakura, A Kawasaki, T Sugasawa - Synthetic Communications, 1988 - Taylor & Francis
Simple Synthesis of 3-Alkyl-1H-Indazoles Having Functional Groups At the ω-Position Page
1 SYNTHETIC COMMUNICATIONS, 18(3), 259-264 (1988) SIMPLE S Y NTH ES 1 S 0 F 3-A …

СИНТЕЗ 3-R2-4-R1-5-АЦЕТИЛ(ЭТОКСИКАРБОНИЛ)-6-ГИДРОКСИ-6-МЕТИЛИНДАЗОЛОВ

ВB Сорокин, АB Григорьев, АK Рамазанов… - Chemistry of …, 1999 - hgs.osi.lv
It was discovered that functionally substituted tetrahydroindazoles can be aromatized by the
action of sulfur. Previously unknown 3-R 2-4-R 1-5-acetyl (ethoxycarbonyl)-6 …

[PDF][PDF] SYNTHESIS OF DIMETHYLPYRAZOL0 [1, 2-aIBENZOTRIAZOLES AND OF METHYLPYRAZOLO [1, 2-aIQUIN0XALINES BY CYCLIZATION OF 3.5-DIMETHYL …

A Albini, G Bettinetti, G Minoli - Heterocycles, 1995 - library.navoiy-uni.uz
--The thermal and photochemical decomposition of a series of 5-substituted I-(2-
azidopheny1)-3.5-dimethylpyrazoles has been examined under a homogeneous set of …

[引用][C] Regioselective Synthesis of 2-N-Substituted 6-Nitro-and 4, 6-Dinitroindazoles

DA Brovko, VN Marshalkin, VV Semenov - Chemistry of Heterocyclic …, 2001 - Springer
2-N-Substituted indazoles can be obtained from N-(2-nitrobenzylidene) amines via
reduction by carbon monoxide in the presence of iron carbonyls [1], and also by treatment …

Synthesis of di-and trisubstituted 1, 2, 4-triazoles containing indole fragments

VI Kelarev, RA Karakhanov, SS Gasanov… - Chemistry of …, 1993 - Springer
The reaction of imino esters of indole-series acids with acid hydrazides gave N (1)-
acylamidrazones, which, during heating, were converted to 3, 5-disubstituted 1H-1, 2, 4 …

Synthesis of 3‐dialkylaminomethyl‐5‐methyl‐4‐substituted‐1H‐pyrazoles. Selective functionalization of one methyl group via n‐nitration of 3, 5‐dimethyl‐4 …

H Lammers, R Vollinga, P Zandbergen… - Journal of …, 1995 - Wiley Online Library
Abstract Treatment of 4‐substituted 3, 5‐dimethyl‐1‐nitro‐1H‐pyrazoles 1 and 10a‐c with
secondary amines in acetonitrile, in the presence of 1, 8‐diazabicyclo [5.4. 0] undec‐7‐ene …

A method for the regioselective synthesis of 1-alkyl-1H-indazoles

HJ Liu, SF Hung, CL Chen, MH Lin - Tetrahedron, 2013 - Elsevier
A method for the regioselective synthesis of 3-unsubstituted 1-alkyl-1H-indazoles, starting
with 2-halobenzonitriles and N-alkylhydrazines, is described. The two-step reaction pathway …