Guaiazulene and related compounds: A review of current perspective on biomedical applications

W Akram, P Tagde, S Ahmed, S Arora, TB Emran… - Life Sciences, 2023 - Elsevier
Background Thousands of people worldwide pass away yearly due to neurological
disorders, cardiovascular illnesses, cancer, metabolic disorders, and microbial infections …

Synthesis and antigastric ulcer activity of novel 5-isoproyl-3, 8-dimethylazulene derivatives

LY Zhang, F Yang, WQ Shi, P Zhang, Y Li… - Bioorganic & medicinal …, 2011 - Elsevier
5-Isoproyl-3, 8-dimethylazulene derivatives were synthesized and evaluated for antigastric
ulcer activity in vivo. Some of them possess the best activity against gastric ulcer with ulcer …

Anti-Helicobacter pylori agents. An update.

EM Muri, JS Williamson - Mini reviews in medicinal chemistry, 2004 - europepmc.org
Helicobacter pylori infection is the major causative factor of a number of gastric pathologies.
Several classes of compounds have been identified as anti-H. pylori agents. Here we …

In vitro anti-Helicobacter pylori activity of BAS-118, a new benzamide derivative

I Kobayashi, H Muraoka, M Hasegawa… - Journal of …, 2002 - academic.oup.com
The antibacterial activity of BAS-118, a new benzamide derivative, against Helicobacter
pylori and other species of bacteria was investigated, as was the in vitro ability of the …

The ultrafast energy transfer process in naphtole–nitrobenzofurazan bichromophoric molecular systems: A study by femtosecond UV–vis pump-probe spectroscopy

PL Gentili, M Mugnai, L Bussotti, R Righini… - … of Photochemistry and …, 2007 - Elsevier
This work presents an experimental and computational study of the intramolecular electronic
energy transfer process occurring in two newly synthesized bichromophoric species: N-(7 …

[HTML][HTML] α-Anilinoketones, Esters and Amides: A Chemical Study

AM Qandil, LI Fakhouri - Pharmaceuticals, 2012 - mdpi.com
A group of α-anilinoketones, 2-aminoalcohols, α-anilinoesters and α-anilinoamides were
successfully synthesized and characterized by NMR spectroscopy and mass spectrometry …

Green synthesis and microcalorimetric study of a novel N-alkylation Schiff base and its bismuth(III) complex

X Li, GY Le, QG Li, JH Jiang, F Zeng, X Li… - Journal of Thermal …, 2022 - Springer
A new N-alkylation Schiff base [N 2, N 6-bis (2-hydroxy-3-methoxybenzyl) pyridine-2, 6-
dicarboxamide] was synthesized from o-vanillin and pyridine-2, 6-dicarboxamide by a solid …

Discovering novel antibacterial agents by high throughput screening

S Donadio, L Brandi, S Serina… - Frontiers in Drug …, 2005 - ingentaconnect.com
The increasing frequency of nosocomial infections due to multiresistant bacterial pathogens
represents a serious health concern and is continuously threatening the therapeutic …

Facile Synthesis of Aryl‐Pyridyl, Pyridazinyl, Pyrazinyl, and Triazinyl Acetonitriles

AA Farahat, DW Boykin - Journal of Heterocyclic Chemistry, 2013 - Wiley Online Library
Dihalo pyridine, pyrazine, and pyridazine analogues were converted to the corresponding
monohalo acetonitrile analogues through nucleophilic displacement of the halogen with the …

Glyoxyl analogs of indole phytoalexins: Synthesis and anticancer activity

P Kutschy, A Sýkora, Z Čurillová… - Collection of …, 2010 - cccc.uochb.cas.cz
Glyoxyl analogs of indole phytoalexins brassinin, 1-methoxybrassinin, brassitin, 1-
methoxybrassitin and 1-methoxybrassenin B were prepared, using (1 H-indol-3-yl)-,(1 …