Pyrazole-based analogs as potential antibacterial agents against methicillin-resistance staphylococcus aureus (MRSA) and its SAR elucidation
Methicillin-resistant Staphylococcus aureus (MRSA) is becoming lethal to humanity due to
easy transmission and difficult-to-treat skin and flimsy diseases. The most threatening aspect …
easy transmission and difficult-to-treat skin and flimsy diseases. The most threatening aspect …
Heterogeneous graphitic carbon nitrides in visible-light-initiated organic transformations
In recent years, g-C3N4 photocatalyst-mediated organic reactions have represented an
important mode of chemical transformations and are expected to become a crucial field at …
important mode of chemical transformations and are expected to become a crucial field at …
Saturated five-membered thiazolidines and their derivatives: from synthesis to biological applications
In past decades, interdisciplinary research has been of great interest for scholars.
Thiazolidine motifs behave as a bridge between organic synthesis and medicinal chemistry …
Thiazolidine motifs behave as a bridge between organic synthesis and medicinal chemistry …
5-Ene-4-thiazolidinones–An efficient tool in medicinal chemistry
The presented review is an attempt to summarize a huge volume of data on 5-ene-4-
thiazolidinones being a widely studied class of small molecules used in modern organic and …
thiazolidinones being a widely studied class of small molecules used in modern organic and …
A key review on oxadiazole analogs as potential methicillin-resistant Staphylococcus aureus (MRSA) activity: Structure-activity relationship studies
Methicillin-resistant Staphylococcus aureus (MRSA) is becoming dangerous to human
beings due to easy transmission mode and leading to the difficult-to-treat situation. The rapid …
beings due to easy transmission mode and leading to the difficult-to-treat situation. The rapid …
Benzimidazole analogues as efficient arsenals in war against methicillin-resistance staphylococcus aureus (MRSA) and its SAR studies
Small molecule based inhibitors development is a growing field in medicinal chemistry. In
recent years, different heterocyclic derivatives have been designed to counter the infections …
recent years, different heterocyclic derivatives have been designed to counter the infections …
Structure-activity relationship studies of thiazole agents with potential anti methicillin-resistance Staphylococcus aureus (MRSA) activity
Due to the increasing resistance of methicillin-resistant Staphylococcus aureus (MRSA) to
conventional antibiotics, further efforts are needed to develop new antimicrobial agents …
conventional antibiotics, further efforts are needed to develop new antimicrobial agents …
Fluorinated azoles as effective weapons in fight against methicillin-resistance staphylococcus aureus (MRSA) and its SAR studies
The rapid spread of Methicillin-resistant Staphylococcus aureus (MRSA) and its difficult-to-
treat skin and filmsy diseases are making MRSA a threat to human life. The most dangerous …
treat skin and filmsy diseases are making MRSA a threat to human life. The most dangerous …
Synthesis and biological evaluation of purine-pyrazole hybrids incorporating thiazole, thiazolidinone or rhodanine moiety as 15-LOX inhibitors endowed with …
OS Afifi, OG Shaaban, HA Abd El Razik, SEDAS El… - Bioorganic …, 2019 - Elsevier
Novel purine-pyrazole hybrids combining thiazoles, thiazolidinones and rhodanines, were
designed and tested as 15-LOX inhibitors, potential anticancer and antioxidant agents. All …
designed and tested as 15-LOX inhibitors, potential anticancer and antioxidant agents. All …
Design, synthesis and biological evaluation of novel pyridine-thiazolidinone derivatives as anticancer agents: Targeting human carbonic anhydrase IX
In order to obtain novel Human carbonic anhydrase IX (CAIX) inhibitors, a series of pyridine-
thiazolidinone derivatives was synthesized and characterized by various spectroscopic …
thiazolidinone derivatives was synthesized and characterized by various spectroscopic …