Indoles are privileged heterocycles found in many biologically active pharmaceuticals and
natural products. However, the selective functionalization of the benzenoid moiety in indoles …

Herein we report the results of a synthetic strategy toward the marine alkaloid convolutindole
A, a structurally remarkable derivative of the hallucinogen N, N-dimethyltryptamine (DMT) …

Indole derivatives are associated with a variety of both biological activities and applications
in the field of material chemistry. A number of different strategies for synthesizing substituted …

We report the first total synthesis of (−)-kopsifoline A and (+)-kopsifoline E. Our synthetic
strategy features a biogenetically inspired regioselective C17-functionalization of a versatile …

Subjecting 6-bromoindole to an iridium-catalysed triborylation-diprotodeborylation
sequence followed by Chan-Evans-Lam coupling gives 6-bromo-4-methoxyindole in good …

Site-selective late-stage functionalizations of a pyrano [3, 2-a] carbazole core related to the
murrayamine natural products is reported. Specifically, selective C3 and C6 bromination has …

A convenient two-step preparation of NH-free 5-aryl-pyrrole-2-carboxylates is described.
The synthetic route consists of catalytic borylation of commercially available pyrrole-2 …

The isolation of evermore complex natural products has been continuously inspiring
chemists to achieve total syntheses of such targets, while pushing the frontiers of the field of …

We report the first total synthesis of (–)-kopsifoline A and (+)-kopsifoline E. Our synthetic
strategy features a biogenetically inspired regioselective C17-functionalization of a versatile …

Herein we report the results of a synthetic strategy toward the marine alkaloid convolutindole
A, a structurally remarkable derivative of the hallucinogen N, N-dimethyltryptamine (DMT) …