Selective Oxidative Decarbonylative Cleavage of Unstrained C(sp3)–C(sp2) Bond: Synthesis of Substituted Benzoxazinones

A Verma, S Kumar - Organic Letters, 2016 - ACS Publications
A transition metal (TM)-free practical synthesis of biologically relevant benzoxazinones has
been established via a selective oxidative decarbonylative cleavage of an unstrained C (sp …

Synthesis, antimicrobial and anti-inflammatory activity of some new benzoxazinone and quinazolinone candidates

MAEA El-Hashash, ME Azab, RAEA Faty… - Chemical and …, 2016 - jstage.jst.go.jp
Benzoxazinones and quinazolinones have a wide spectrum of biological activity. In this
paper we focused on studying the antimicrobial and anti-inflammatory activities of some …

Rotational Behavior about the N3–Pyridyl Bond in 3-(Pyridin-2-yl) quinazolin-4-one and 4-Thione Derivatives

Y Wang, Y Yang, D Homma, E Caytan… - The Journal of …, 2024 - ACS Publications
The rotational barriers about the N3–(2-pyridyl) bond in 2-iso-propyl-3-(pyridin-2-yl)
quinazolin-4-one and the thione analogue were evaluated though VT-NMR measurement of …

[PDF][PDF] Efficient and convenient route to the synthesis of some novel sulfonate ester-based heterocycles as antitumor agents

A El-Mekabaty, OMO Habib, MA El-Moneim… - …, 2018 - triggered.edina.clockss.org
In the present investigation, simple and straightforward methodology for the preparation of
novel thiazolidinone, thiazole, pyridinone, chromene, pyrazole, benzimidazo [1, 2-a] …

Facile Route for synthesis of novel flame retardant, reinforcement and antibacterial textile fabrics coatings

NF Attia, MH Soliman, SS El-Sakka - Coatings, 2020 - mdpi.com
New and innovative textile fabrics coatings were facilely developed. The coating was
developed based on synthesis of novel charring and antibacterial organic agent in …

Insilco design and potential cytotoxic agents EGFR inhibitors of 4 (3h) quinazolinone derivatives

K Kavitha, N Srinivasan, S Mohan… - Research Journal of …, 2021 - indianjournals.com
Epidermal growth factor receptor (EGFR) acting very important part in cell growth regulation,
one of the most significant consideration studied targets of tyrosine kinases (TK) inhibitors. A …

Synthesis of Novel pyrimido [4, 5-b] quinoline-4-one Derivatives and Assessment as Antimicrobial and Antioxidant Agents

U Fathy, RS Gouhar, A Younis… - Pharmacognosy …, 2021 - phcogj.com
Objective: Antimicrobial resistance has emerged as one of the serious global health
problems of the 21 st century that threatens the efficient treatment and prevention of an …

Evaluation of newly synthesized quinazolinone derivatives of hydrazones as potent anti-inflammatory and antibacterial agents

B Kandpal, J Meshram, I Mohanram… - Medicinal Chemistry …, 2015 - Springer
The present work describes the newly synthesized series of 4-(3H)-quinazolinone
derivatives of hydrazones 5 (a–j) starting from benzoxazine (4) by conventional method and …

[PDF][PDF] Synthesis, molecular docking study and brine shrimp lethality test of benzoxazine and aminomethyl derivatives from eugenol

GS Putra, TA Yuniarta, A Syahrani… - International Journal of …, 2016 - researchgate.net
The specific objective of this research is to study the reaction of eugenol with formaldehyde
and aniline and to perform in silico and biological activity studies on the obtained products …

Recyclable Keggin Heteropolyacids as an Environmentally Benign Catalyst for the Synthesis of New 2-Benzoylamino-N-phenyl-benzamide Derivatives under …

K Ighilahriz-Boubchir, B Boutemeur-Kheddis, C Rabia… - Molecules, 2017 - mdpi.com
2-Benzoylamino-N-phenyl-benzamide derivatives (5a–h) were prepared from 2-phenyl-3, 1-
(4 H)-benzoxazin-4-one 3 and substituted anilines 4a–h in the presence of a Keggin-type …