[HTML][HTML] Antimicrobial activities of heterocycles derived from thienylchalcones

O Mazimba - Journal of King Saud University-Science, 2015 - Elsevier
Thiophene analogues of chalcones were synthesized in good yields by condensation of 2-
acetylthiophene and salicylaldehydes. Solvent-free Michael addition of cyclohexanone to 2 …

In Vitro Cytotoxicity and Aromatase Inhibitory Activity of Flavonoids: Synthesis, Molecular Docking and In Silico ADME Prediction

U Shah, S Patel, M Patel, N Jain… - Anti-Cancer Agents …, 2022 - ingentaconnect.com
Background: Many natural and synthetic flavonoids have been studied and documented by
inhibiting aromatase enzymes for their anti-cancer activity against breast carcinoma. The …

Synthesis of 1, 3-diaryl-2-propene-1-one derivatives using Tripotassium phosphate as an alternative and efficient catalyst and study its cytotoxic and antimicrobial …

P Patil, P Khan, S Zangade - Current Chemistry Letters, 2020 - m.growingscience.com
A series of fourteen chalcone was synthesized via. Claisen–Schmidt condensation between
substituted 2-hydroxyl acetonaphthones and substituted benzaldehyde in presence of …

Alumina-K3PO4 solid supported microwave synthesis of 1, 3-diaryl-2-propene-1-one derivatives as a prominent antioxidant scavenger

P Patil, G Bhopalkar, S Zangade - Current Microwave …, 2020 - ingentaconnect.com
Background: The various industrial processes have a diverse effect on the environment
through pollution. In view of these observations, some environmentally benign synthetically …

[PDF][PDF] Synthesis of Substituted Chalcones and Investigation of Their Biological Activities

SA Rashdan, AM Hassan, QA Mandeel… - Journal of …, 2018 - jcb.thebrpi.org
The synthesis of highly antioxidants and antimicrobial agents has attracted great attention
due to their high importance to human health. Chalcones are known to exhibit wide …

[HTML][HTML] Sintesis Senyawa Basa Schiff dari Vanilin dan p-Aminoasetofenon dengan menggunakan Katalis Asam Alami Jus Jeruk Nipis serta pemanfaatannya sebagai …

L Ma'rufah - 2020 - etheses.uin-malang.ac.id
مستخلص البحث مركب قلوي شيف يوجد هغا شيف فى السنة ١٨٦٤. قلوي شيف يستطيع أن يوليف
من المركب الأمينية الأولية الذي يتفاعل مع الأدهيد أو الكيتون. مركب قلوي شيف المعروف باسم …

Variasi Mol Katalis NaOH pada sintesis senyawa turunan kalkon dari vanilin dan asetofenon menggunakan metode penggerusan

A Srilistiani - 2019 - etheses.uin-malang.ac.id
INDONESIA: Sintesis senyawa yang sesuai dengan prinsip green chemistry dinamakan
green-synthesis, salah satunya adalah teknik penggerusan yang memberikan waktu relatif …

Sintesis Senyawa 1, 5-bis (4-hidroksi-3-metoksifenil) penta-1, 4-dien-3-on dengan Variasi Mol NaOH Melalui Reaksi Kondensasi Claisen-Schmidt Menggunakan …

F Farchana - 2016 - etheses.uin-malang.ac.id
INDONESIA: Sintesis senyawa yang sesuai dengan prinsip green chemistry dinamakan
green-synthesis, salah satunya adalah teknik penggerusan yang memberikan waktu reaksi …

Sintesis senyawa 1, 5-bis (4-hidroksi-3-metoksifenil) penta-1, 4-dien-3-on melalui kondensasi claisen-schmidt dengan variasi mol vanilin teknik penggerusan

C Ulum - 2016 - etheses.uin-malang.ac.id
INDONESIA: Senyawa vanilin memiliki aktivitas antikanker yang lemah dengan nilai IC50
sebesar 1.360, 17 µg/mL. Modifikasi struktur vanilin dilakukan untuk meningkatkan aktivitas …

[PDF][PDF] International Journal for Pharmaceutical Research Scholars (IJPRS)

SB Shaikh, S Mujahid, N Tambat, K Salgar… - researchgate.net
ABSTRACT Chalcones have characteristic 1, 3-diaryl-2-propen-1-one backbone skeleton.
Changes in their aryl ring have offered a high degree of diversity that has proven useful for …