1, 2-Amino alcohols and their heterocyclic derivatives as chiral auxiliaries in asymmetric synthesis

DJ Ager, I Prakash, DR Schaad - Chemical Reviews, 1996 - ACS Publications
R-amino acid reductions, allow entry to other classes of compounds that are also useful as
the source of chiral centers, as with R-amino aldehydes, that, in turn, can be used in a …

A convenient reduction of amino acids and their derivatives

MJ McKennon, AI Meyers, K Drauz… - The Journal of Organic …, 1993 - ACS Publications
A convenient reduction of amino acids and their derivatives Page 1 3568 J. Org. Chem. 1993,58,
3568-3571 A Convenient Reduction of Amino Acids and Their Derivatives Marc J. McKennon …

Triurethane-protected guanidines and triflyldiurethane-protected guanidines: new reagents for guanidinylation reactions

K Feichtinger, HL Sings, TJ Baker… - The Journal of …, 1998 - ACS Publications
New guanidinylation reagents are reported. These reagents consist of N, N ', N ''-tri-Boc-
guanidine (1) and N, N ', N ''-tri-Cbz-guanidine (2), which allow for the facile conversion of …

Design and Synthesis of Cyclopenta[g]quinazoline-Based Antifolates as Inhibitors of Thymidylate Synthase and Potential Antitumor Agents,

V Bavetsias, JH Marriott, C Melin… - Journal of medicinal …, 2000 - ACS Publications
Following the development of raltitrexed, the synthesis of nonpolyglutamatable inhibitors of
TS that do not use the reduced folate carrier (RFC) for cellular entry should provide …

[图书][B] Combinatorial peptide and nonpeptide libraries: a handbook

G Jung - 2008 - books.google.com
Millionen von Peptiden, sogenannte Peptidbibliotheken, simultan, schnell und oft auch
schon automatisiert herzustellen, gelingt mit der kombinatorischen Chemie. Diese …

Mild reduction of carboxylic acids to alcohols using cyanuric chloride and sodium borohydride

M Falorni, A Porcheddu, M Taddei - Tetrahedron letters, 1999 - Elsevier
Mild Reduction of Carboxylic Acids to Alcohols Using Cyanuric Chloride and Sodium
Borohydride Page 1 Pergamon Tetrahedron Letters 40 (1999) 4395-4396 TETRAHEDRON …

Improvement of Pharmacokinetics of Radioiodinated Tyr3-Octreotide by Conjugation with Carbohydrates

M Schottelius, HJ Wester, JC Reubi… - Bioconjugate …, 2002 - ACS Publications
Among a variety of other factors, the clearance kinetics and routes of excretion of
radiopharmaceuticals are of crucial importance for early and high tumor/background ratios …

Short synthesis of (+)-Cylindricine C by using a catalytic asymmetric Michael reaction with a two-center organocatalyst

T Shibuguchi, H Mihara… - Angewandte …, 2006 - kyushu-u.elsevierpure.com
Abstract (Chemical Equation Presented) Two for the price of one: The total synthesis of (+)-
cylindricine C has been achieved in six steps using a catalytic asymmetric Michael reaction …

Inhibition of Group IVA Cytosolic Phospholipase A2 by Novel 2-Oxoamides in Vitro, in Cells, and in Vivo

G Kokotos, DA Six, V Loukas, T Smith… - Journal of medicinal …, 2004 - ACS Publications
The Group IVA cytosolic phospholipase A2 (GIVA PLA2) is a particularly attractive target for
drug development because it is the rate-limiting provider of proinflammatory mediators. We …

[PDF][PDF] Effective and mild method for preparation of optically active α-amino aldehydes via TEMPO oxidation

J Jurczak, D Gryko, E Kobrzycka, H Gruza… - Tetrahedron, 1998 - academia.edu
The TEMPO oxidation method is successfully applied to preparation of variously protected,
optically active ct-amino aldehydes without racemization and in very good yield.© 1998 …