Hydrazides/hydrazones as antimicrobial and anticancer agents in the new millennium

P Kumar, B Narasimhan - Mini reviews in medicinal chemistry, 2013 - ingentaconnect.com
Hydrazide/hydrazone derivatives are of quite interest for medicinal chemists because of their
vast spectrum of biological activity. Literature reports reveal that the hydrazide derivatives …

Design, synthesis, antimicrobial, anticancer evaluation, and QSAR studies of 4-(substituted benzylidene-amino)-1, 5-dimethyl-2-phenyl-1, 2-dihydropyrazol-3-ones

S Sigroha, B Narasimhan, P Kumar, A Khatkar… - Medicinal Chemistry …, 2012 - Springer
A series of 4-(substituted benzylidene-amino)-1, 5-dimethyl-2-phenyl-1, 2-dihydropyrazol-3-
ones (1–17) was synthesized and tested in vitro for its antimicrobial and anticancer …

[PDF][PDF] Biological prospective of 4-thiazolidinone: a review

R Kumar, S Patil - Hygeia: Journal for Drugs and Medicines, 2017 - hygeiajournal.com
Plan: Biological prospective of 4-thiazolidinone Prologue: 4-Thiazolidinones are derivatives
of thiazolidine with a carbonyl group in the 4th position. Substitution on the 2nd, 3rd and 5th …

Novel thiazolidinone-containing compounds, without the well-known sulphonamide zinc-binding group acting as human carbonic anhydrase IX inhibitors

Ö Güzel-Akdemir, A Angeli, K Demir… - Journal of Enzyme …, 2018 - Taylor & Francis
A small collection of 26 structurally novel thiazolidinone-containing compounds, without the
well-known sulphonamide zinc-binding group, were synthesised and tested in enzyme …

Synthesis of novel imidazo [1, 2-a] pyridines and evaluation of their antifungal activities

F GÖKTAŞ, N Cesur, D ŞATANA… - Turkish Journal of …, 2014 - journals.tubitak.gov.tr
Abstract New 2-(imidazo [1, 2-a] pyridin-2-ylcarbonyl)-N-substituted
hydrazinecarbothioamides (4a--j), N'-(3-substituted-4-oxo-1, 3-thiazolidin-2-ylidene) imidazo …

[HTML][HTML] Synthesis and aldose reductase inhibitory effect of some new hydrazinecarbothioamides and 4-thiazolidinones bearing an imidazo [2, 1-b] thiazole moiety

NU Güzeldemirci, S Cimok, DAŞE Net… - Turkish Journal of …, 2019 - ncbi.nlm.nih.gov
Objectives: To synthesize and characterize 2-[[6-(4-bromophenyl) imidazo [2, 1-b] thiazol-3-
yl] acetyl]-N-alkyl/arylhydrazinecarbothioamide and 3-alkyl/aryl-2-[((6-(4-bromophenyl) …

[HTML][HTML] N-[2-(4-Chlorophenyl)-5-methyl-4-oxo-1, 3-thiazolidin-3-yl] pyridine-3-carboxamide

M Akkurt, I Celik, H Demir, S Özkırımlı… - … Section E: Structure …, 2011 - scripts.iucr.org
The title compound, C16H14ClN3O2S, crystallizes with two molecules in the asymmetric
unit. In the 1, 3-thiazolidine rings, the carbonyl O atoms, the S atoms, the methyl groups and …

[HTML][HTML] Synthesis and antimicrobial activities of some new azetidin-2-ones and thiazolidin-4-ones

SR Desai, UV Laddi, RS Bennur… - Indian journal of …, 2011 - ncbi.nlm.nih.gov
Abstract Various (4-substituted) phenyl-3-β-[(N-benzenesulphonyl/tosyl)-4-(un) substituted
anilino] propionylamido-1, 3-thiazolidine-4-ones (3a–x) and 1-β-[(N-benzenesulphonyl/tosyl …

Regioselective Synthesis of Novel 3‐Thiazolidine Acetic Acid Derivatives from Glycosido Ureides

Y Li, W Chen, X Yang, G Yu, M Mao… - Chemical Biology & …, 2011 - Wiley Online Library
A series of 3‐thiazolidine acetic acid‐2‐(per‐O‐acetylglycosyl)‐1′‐imino‐α‐(substituted)‐4‐
oxo ethyl ester derivatives (3a–t) were prepared via the reaction of substituted amino acid‐N …

[PDF][PDF] İMİDAZO [2, 1-b] TİYAZOL TÜREVİ BAZI TİYAZOLİDİNONLARIN

SVE KARAKTERİZASYONLARI, M İSAOĞLU… - nek.istanbul.edu.tr
Bu tez çalışmasının kendi çalışmanı olduğunu, Lczin planlanmasından yazımına kadar
bütün sathal ıırda etik d ı şı davran ı şımın ol madığını, bu tezdeki biltOıı bilgileri akademik ve …