Primaquine revisited six decades after its discovery
Primaquine was firstly synthesized in 1946 in the USA, and is the most representative
member of the anti-malarial 8-aminoquinolines. Six decades have passed and primaquine …
member of the anti-malarial 8-aminoquinolines. Six decades have passed and primaquine …
8-Aminoquinolines: future role as antiprotozoal drugs
BL Tekwani, LA Walker - Current opinion in infectious diseases, 2006 - journals.lww.com
Extensive derivatization approaches followed by better understanding of structure-activity
relationships and biotransformation mechanisms of toxicity have provided 8-aminoquinoline …
relationships and biotransformation mechanisms of toxicity have provided 8-aminoquinoline …
Imidazoquines as antimalarial and antipneumocystis agents
Peptidomimetic imidazolidin-4-one derivatives of primaquine (imidazoquines) recently
displayed in vitro activity against blood schizonts of a chloroquine-resistant strain of …
displayed in vitro activity against blood schizonts of a chloroquine-resistant strain of …
Anti-Pneumocystis carinii and antiplasmodial activities of primaquine-derived imidazolidin-4-ones
A series of primaquine-derived imidazolidin-4-ones were screened for their in vitro activity
against Pneumocystis carinii and Plasmodium falciparum W2 strain. Most compounds were …
against Pneumocystis carinii and Plasmodium falciparum W2 strain. Most compounds were …
[引用][C] Νέοι υβριδικοί παράγοντες αρτεμισινίνης και πριμακίνης με πιθανή αντικαρκινική και ανθελονοσιακή δράση
Χ Αβραάμ - 2021