[HTML][HTML] Thiazole ring-the antimicrobial, anti-inflammatory, and anticancer active scaffold

S Hosseininezhad, A Ramazani - Arabian Journal of Chemistry, 2023 - Elsevier
Background Thiazole ring is one of the most important heterocycle scaffolds in organic and
medicinal chemistry due to this scaffold being the backbone of numerous drugs and their …

Recent updates on the synthesis of thiazolopyrimidines derivatives

MS Nazir, S Aslam, M Ahmad… - Synthetic …, 2023 - Taylor & Francis
Fused heterocyclic ring structures play an important role in the enhancement of
pharmaceutical actions of the molecules and have been reported to have efficient medicinal …

[HTML][HTML] Synthesis, characterization, and biological investigations of potentially bioactive heterocyclic compounds containing benzimidazole nucleus

R Champa, KA Vishnumurthy, YD Bodke, HSB Naik… - Results in …, 2023 - Elsevier
Six benzimidazole derivatives have been synthesized and characterized using
spectroscopic techniques such as IR, 1 H NMR, 13 C NMR, and mass spectrometry. The …

An efficient p‐TSA catalyzed synthesis of some new substituted‐(5‐hydroxy‐3‐phenylisoxazol‐4‐yl)‐1, 3‐dimethyl‐1H‐chromeno [2, 3‐d] pyrimidine‐2, 4 (3H, 5H) …

SH Sukanya, T Venkatesh, SJA Rao… - Journal of Molecular …, 2022 - Elsevier
We have developed an easy and efficient protocol for the synthesis of a series of some novel
substituted-(5-hydroxy-3-phenylisoxazol-4-yl)-1, 3-dimethyl-1H-chromeno [2, 3-d] pyrimidine …

(2-Hydroxy-3-Methoxybenzylidene)thiazolo[3,2-a]pyrimidines: Synthesis, Self-Assembly in the Crystalline Phase and Cytotoxic Activity

AS Agarkov, AA Nefedova, ER Gabitova… - International Journal of …, 2023 - mdpi.com
A series of new 2-hydroxy-3-methoxybenzylidenethiazolo [3, 2-a] pyrimidines with different
aryl substituents at the 5 position are synthesized and characterized by 1H/13C NMR and IR …

One-pot synthesis of some new 7‑hydroxy-5-(4-substitutedphenyl)-9-methyl-1, 5-dihydro-2H-dipyrimido [1, 2-a: 4′, 5′-d] pyrimidine-2, 4 (3H)‑dione derivatives and …

K Upendranath, T Venkatesh, M Shashank… - Journal of Molecular …, 2022 - Elsevier
Metal-free organic dyes are gaining interest and demands in the field of light absorption and
light-emitting applications. In this study, we developed efficient one-pot synthesis of 7 …

L-Proline: Unraveling its Reactivity and Mechanistic Insights as an Organocatalyst in Multi-Component Synthesis: A Comprehensive Review

BS Saikia, I Rahman, P Nath, A Boruah, ML Deb… - Catalysis …, 2024 - Taylor & Francis
ABSTRACT L-Proline has emerged as a cornerstone in organocatalysis, celebrated for its
versatility and efficiency in promoting a wide range of chemical transformations. This review …

Synthesis, Self-Assembly in Crystalline Phase and Anti-Tumor Activity of 2-(2-/4-Hydroxybenzylidene)thiazolo[3,2-a]pyrimidines

AS Agarkov, AA Nefedova, ER Gabitova… - Molecules, 2022 - mdpi.com
A series of new thiazolo [3, 2-a] pyrimidines different by aryl substituents in 2 and 5 positions
are synthesized and characterized in solution as well as in the crystalline phase using 1H …

Water mediated pot, atom, and step economic (PASE) synthesis of pyrimido[4,5-d]pyrimidines using ultrasound and microwave irradiation approaches

HD Trivedi, VB Joshi, BY Patel - Synthetic Communications, 2023 - Taylor & Francis
Abstract The functioning, Pot, Atom, and Step Economic (PASE) green chemistry proposition
has been approached for the synthesis of pyrimido [4, 5-d] pyrimidines by the …

Synthesis, Structure, and In Vitro Pharmacological Evaluation of some New Pyrimidine-2-Sulfonamide Derivatives and Their Molecular Docking Studies on Human …

QAH Jaber, AH Shentaif, M Almajidi, I Ahmad… - Russian Journal of …, 2023 - Springer
In this approach, novel pyrimidine-2-sulfonamide derivatives based on the 2 H-chromen-2-
one moiety were synthesized and evaluated as anticancer and antibacterial agents …