From Bench to Bedside: What Do We Know about Imidazothiazole Derivatives So Far?

M Guo, X Yu, YZ Zhu, Y Yu - Molecules, 2023 - mdpi.com
Imidazothiazole derivatives are becoming increasingly important in therapeutic use due to
their outstanding physiological activities. Recently, applying imidazothiazole as the core …

[PDF][PDF] Synthesis, docking study and in vitro anticancer evaluation of new derivatives of 2-(1-(2-flouro-[1, 1-biphenyl]-4-yl) ethyl)-6-(substituted phenyl) imidazole [2, 1-B …

KS Hmood, AARM Kubba - Systematic Reviews in Pharmacy, 2020 - academia.edu
Results: The new compounds were characterized by FTIR, 1HNMRs and CHNS analysis. A
molecular docking study of the synthesized compounds (2-5) against HIV protease indicated …

[PDF][PDF] Synthesis, and Anti-Tumor Evaluation of Some New Flurbiprofen Derivatives against MCF-7 and WRL-68 Cell Lines.

KS Hmood, AAR Mahmood Kubba… - Indonesian Journal of …, 2021 - core.ac.uk
(VEGFR-2) was applied, and it indicated that compounds 4, 7, 13, and 15, exhibited the
optimum binding energy of-6.77,-6.12,-6.68,-6.43 kcal/mol, respectively. Target compounds …

[HTML][HTML] Ornidazole Reduces the progression of endometriosis in a rat model

X Qin, H Yang, D Qiao, X Liu, LB Liu, SF Liu… - Gynecologic and …, 2022 - karger.com
Objective: The aim of this study was to investigate the effectiveness of ornidazole in
inhibiting the progression of endometriosis in a rat model. Design: This was an in vivo …

Synthesis, Molecular Docking Studies and ADME Prediction of Some New Albendazole Derivatives as α-Glucosidase Inhibitors.

S Şenkardeş, N Kulabaş… - Acta Chimica …, 2022 - search.ebscohost.com
A series of novel 2-(substituted arylidene)-N-(5-(propylthio)-2, 3-dihydro-1H-benzo [d]
imidazol-2-yl) hydrazine-1-carboxamide derivatives 3a–i were synthesized via condensation …

Synthesis, Molecular Docking Studies and ADME Prediction of Some New Albendazole Derivatives as α-Glucosidase Inhibitors.

S Senkardes, N Kulabas, SG Kucukguzel - Acta Chimica Slovenica, 2022 - europepmc.org
A series of novel 2-(substituted arylidene)-N-(5-(propylthio)-2, 3-dihydro-1H-benzo [d]
imidazol-2-yl) hydrazine-1-carboxamide derivatives 3a-i were synthesized via condensation …

[PDF][PDF] Synthesis, Characterization, and Antimicrobial Evaluation for New Azo-linked Derivative of Heterocyclic Compounds.

AA Shafeeq, ZMA Hamandi, MH Mohammed… - Journal of Contemporary …, 2022 - iasj.net
Objectives: Using different activated heterocyclic amines to prepare diazonium salts to be
coupled with ornidazole (heterocyclic agent) to form the azo linkage compounds (A1, A2) as …