Reactions of thioamide dianions, derived from secondary N-arylmethyl thioamides using
BuLi, with thioformamides followed by the addition of iodine to yield 5-amino-2-thiazolines …

Tiazofurin analogues bearing a 5-hydroxymethyl-2-methyl-tetrahydrofuro [2, 3-d][1, 3] dioxol-
6-ol moiety as a sugar mimic (2 and 3), and two novel thiazole-based acyclo-C-nucleosides …

Novel syntheses of C-nucleoside analogs with aryl quinoxalines as nucleobase surrogates
have been accomplished by mild and efficient three-component sequential reactions in high …

Synthesis of three tiazofurin (1) isosteres with nitrogen functionalities at the C-2′ position
(N 3, NH 2 and NH 3+ Cl−) has been achieved, in multistep sequences, starting from …

2-Deoxy-C-nucleosides are a subcategory of C-nucleosides that has not been explored
extensively, largely because the synthesis is less facile. Flexible synthetic procedures giving …

Several reviews dealing with C‐nucleosides covering biological applications and synthetic
methods have been published. This chapter focuses on the chemical synthetic procedures …

A two-step process for the transformation of readily available carbohydrate derivatives into
acyclic C-nucleosides is described. The carbohydrate undergoes a scission process that is …

The synthesis of C-3-substituted het (aryl) indole C-nucleoside analogues bearing
structurally diverse sugar moieties has been achieved by Sonogashira coupling of terminal …

This review will describe the recent advances in the synthesis of C-nucleosides with
inhibitory activity of inosine monophosphate dehydrogenase (IMPDH), a key enzyme in the …

Synthesis of four new tiazofurin analogues has been accomplished starting from d-glucose.
The key step of the synthesis was the three-step cascade that enabled an efficient hydrogen …