In-silico design novel phenylsulfonyl furoxan and phenstatin derivatives as multi-target anti-cancer inhibitors based on 2D-QSAR, molecular docking, dynamics and …

A Guendouzi, L Belkhiri, F Djelti, ZM Zendaoui… - Molecular …, 2024 - Taylor & Francis
ABSTRACT A series of 31 hybrid of phenylsulfonyl furoxan and phenstatin (1a-j, 2a-j, 3a-j, 4
and 5) derivatives, were computationally studied as potential anti-cancer inhibitors against …

[PDF][PDF] QSAR study of benzylidene hydrazine benzamides derivatives with in vitro anticancer activity against human lung cancer cell line A459

GS Putra, MI Sulistyowaty, TA Yuniarta… - Journal of Pharmacy & …, 2023 - academia.edu
Context: In the last decade, resistance to epidermal growth factor receptor-tyrosine kinase
inhibitors (EGFR-TKIs) in lung cancer cases has been widespread. The discovery and …

Synthesis, ADMET predictions, molecular docking studies, and in-vitro anticancer activity of some benzoxazines against A549 human lung cancer cells

MI Sulistyowaty, R Widyowati, GS Putra… - Journal of Basic and …, 2021 - degruyter.com
Objectives This study aims to synthesize a series of benzoxazines (1–5) to be examined as
an epidermal growth factor receptor (EGFR) inhibitor by in-silico study. The overexpression …

N-(2-(2-Benzilidenehydrazinecarbonyl) phenyl) benzamides: Synthesis, Cytotoxic, Antioxidant Activity and Molecular Docking Studies

MI Sulistyowaty, GS Putra, W Zhichao… - Journal of Hunan …, 2020 - repository.unair.ac.id
This study's purpose was to continue our research by acquiring novel anticancer candidates,
the derivatives of N-(2-(2-benzylidenehydrazinecarbonyl) phenyl) benzamide. The …

Immunomodulatory and Anticancer Activities of Barley Bran Grown in Jordan: An in vitro and in vivo Study

SF Abuarab, WH Talib - Frontiers in Nutrition, 2022 - frontiersin.org
The Mediterranean diet is regarded as one of the most healthful dietary patterns in the world,
owing to a combination of foods high in antioxidants and anticancer constituents. Barley …

[HTML][HTML] Benzylidene hydrazine benzamide derivatives QSAR study

Context: In the last decade, resistance to epidermal growth factor receptor-tyrosine kinase
inhibitors (EGFR-TKIs) in lung cancer cases has been widespread. The discovery and …

[PDF][PDF] Journal of Basic and Clinical Physiology and Pharmacology

U Oliviero, AM Marra, G Bosso, E Biskup… - 2022 - researchgate.net
Abstract Objectives: Native Bacillus thuringiensis BK5. 2, isolated from soil of Baluran
National Park, East Java, Indonesia, has been shown to be toxic against Aedes aegypti …