Nucleoside analogues as chemotherapeutic agents: a review
C Périgaud, G Gosselin, JL Imbach - Nucleosides & nucleotides, 1992 - Taylor & Francis
Nucleoside Analogues as Chemotherapeutic Agents: A Review Page 1 NUCLEOSIDES AND
NUCLEOTIDES, 1 1 ( 2 - 4 ) , 9 0 3 - 9 4 5 ( 1 9 9 2 ) NUCLEOSIDE ANALOGUES AS …
NUCLEOTIDES, 1 1 ( 2 - 4 ) , 9 0 3 - 9 4 5 ( 1 9 9 2 ) NUCLEOSIDE ANALOGUES AS …
Adenosine receptors and their modulators
The identification and characterization of adenosine receptors and the development of
potent, receptor subtype-selective agonist and antagonists has been an active area of …
potent, receptor subtype-selective agonist and antagonists has been an active area of …
Anodic benzylic C (sp 3)–H amination: unified access to pyrrolidines and piperidines
S Herold, D Bafaluy, K Muñiz - Green Chemistry, 2018 - pubs.rsc.org
An electrochemical aliphatic C–H amination strategy was developed to access the important
heterocyclic motifs of pyrrolidines and piperidines within a uniform reaction protocol. The …
heterocyclic motifs of pyrrolidines and piperidines within a uniform reaction protocol. The …
N6-Substituted adenosine derivatives: selectivity, efficacy, and species differences at A3 adenosine receptors
ZG Gao, JB Blaustein, AS Gross, N Melman… - Biochemical …, 2003 - Elsevier
The activation of the human A3 adenosine receptor (AR) by a wide range of N6-substituted
adenosine derivatives was studied in intact CHO cells stably expressing this receptor …
adenosine derivatives was studied in intact CHO cells stably expressing this receptor …
Asymmetric electrophilic fluorination using an anionic chiral phase-transfer catalyst
V Rauniyar, AD Lackner, GL Hamilton, FD Toste - Science, 2011 - science.org
The discovery of distinct modes of asymmetric catalysis has the potential to rapidly advance
chemists' ability to build enantioenriched molecules. As an example, the use of chiral cation …
chemists' ability to build enantioenriched molecules. As an example, the use of chiral cation …
Rhodium‐Catalyzed Asymmetric Hydrogenation of 3‐Benzoylaminocoumarins for the Synthesis of Chiral 3‐Amino Dihydrocoumarins
Y Xu, D Liu, Y Deng, Y Zhou… - Angewandte Chemie …, 2021 - Wiley Online Library
An asymmetric hydrogenation of 3‐benzoylaminocoumarins was achieved for the first time
using our BridgePhos‐Rh catalytic system, providing chiral 3‐amino dihydrocoumarins in …
using our BridgePhos‐Rh catalytic system, providing chiral 3‐amino dihydrocoumarins in …
Mast cell degranulation following adenosine A3 receptor activation in rats
JR Fozard, HJ Pfannkuche, HJ Schuurman - European journal of …, 1996 - Elsevier
The present studies were carried out to provide further evidence for the hypothesis that the
hypotensive response to adenosine A3 receptor activation in the anaesthetized rat involves …
hypotensive response to adenosine A3 receptor activation in the anaesthetized rat involves …
Part II: nitroalkenes in the synthesis of heterocyclic compounds
This part (part II) is devoted to 6-membered heterocycles that are synthesized from
nitroalkenes as the key substrates. These compounds can be simply accessible to form …
nitroalkenes as the key substrates. These compounds can be simply accessible to form …
Neuroprotective Principles from Gastrodia elata
Serum deprivation-induced neuronal-like PC12 cell apoptosis was used as an
ischemic/hypoxic model to screen neuroprotective compounds from the rhizomes of …
ischemic/hypoxic model to screen neuroprotective compounds from the rhizomes of …
Exploring distal regions of the A3 adenosine receptor binding site: sterically constrained N6-(2-phenylethyl) adenosine derivatives as potent ligands
S Tchilibon, SK Kim, ZG Gao, BA Harris… - Bioorganic & medicinal …, 2004 - Elsevier
We synthesized phenyl ring-substituted analogues of N6-(1S, 2R)-(2-phenyl-1-cyclopropyl)
adenosine, which is highly potent in binding to the human A3AR with a Ki value of 0.63 nM …
adenosine, which is highly potent in binding to the human A3AR with a Ki value of 0.63 nM …