A spectrum of compounds attached to 2‐keto aryl azole moieties are found as pivotal
building blocks in medicinal chemistry and drug discovery. This is why, the collection of …

A combination of experimental and computational studies have identified a C= O⋅⋅⋅
isothiouronium interaction as key to efficient enantiodiscrimination in the kinetic resolution of …

Molecular iodine in combination with TBHP offers an advanced concept for organic
synthesis and catalysis by improving the selectivity and sustainability of organic …

A novel palladium‐catalyzed C H double carbonylation introduces two adjacent carbonyl
groups for the synthesis of isatins from readily available anilines. The reaction proceeds …

2′-Aminoacetophenones undergo a C (sp3)–H oxidation followed by intramolecular C–N
bond formation by virtue of a simple electrochemical oxidation in the presence of n-Bu4NI …

A novel method toward synthesis of sulfonamides and β-arylsulfonyl enamines has been
developed via I2/TBHP mediated C–N and C–H bond cleavage of tertiary amines, which …

A novel approach for the synthesis of a variety of polysubstituted trans-2, 3-dihydropyrroles
from a wide range of chalcones and β-enamine ketones (esters) via iodine-promoted …

To achieve the goal of green chemistry and sustainable development, catalyst-free reactions
and use of naturally abundant resources are gaining importance. In last two decades, C–H …

Direct C–H functionalization of quinones with arylboronic acids is achieved using K2S2O8
as the sole and efficient green catalytic system. This method provides a straightforward and …

An I2/TBHP-mediated intramolecular dehydrogenative coupling reaction is developed for
the synthesis of a library of medicinally important 5, 11-dialkylindolo [3, 2-c] quinoline salts …