Biannual Account of Anti‐malarial Agents reported in 2021 and 2022: A Comprehensive Coverage

TM Dhameliya, DS Patel, D Kathuria, MB Shah… - …, 2024 - Wiley Online Library
Malaria remains a severe infectious disease caused by Plasmodium parasites among the
primarily afflicting impoverished populations. According to World Health Organization (WHO) …

Proposition of In silico Pharmacophore Models for Malaria: A Review

NF de Sousa, IMA de Araújo… - … Chemistry & High …, 2024 - benthamdirect.com
In the field of medicinal chemistry, the concept of pharmacophore refers to the specific
region of a molecule that possesses essential structural and chemical characteristics for …

Synthesis of Diethyl 6-Amino-1,4-diaryl-2-oxo-1,2,3,4-tetrahydropyridin-3,5-dicarboxylates Based on the Reaction of Arylmethylidenecyanoacetic Esters with N …

KA Avagyan, MS Sargsyan, AE Badasyan… - Russian Journal of …, 2023 - Springer
The reaction of arylmethylidenecyanoacetic esters with N-arylamides of malonic acid led to
the formation of previously unknown diethyl 6-amino-1, 4-diaryl-2-oxo-1, 2, 3, 4 …

New thiazole, thiophene and 2-pyridone compounds incorporating dimethylaniline moiety: synthesis, cytotoxicity, ADME and molecular docking studies

HM Metwally, NM Younis, E Abdel-Latif, A El-Rayyes - BMC chemistry, 2024 - Springer
Various sets of thiazole, thiophene, and 2-pyridone ring structures containing a
dimethylaniline component were synthesized. Substituted thiazoles 2–3 and thiophenes 5–7 …

Synthesis and Characterisation of Amino Functionalised Mesoporous Silica-based Nanomaterials for Isoniazid Drug Delivery

JO Tella, KO Ajanaku, JA Adekoya… - … and Business for …, 2024 - ieeexplore.ieee.org
It was an established norm that conventional drug delivery modules such as tablets and
capsules are prone to poor bioavailability. Hence, in this study, mesoporous silica …