[HTML][HTML] Ultrasound-assisted one-pot green synthesis of new N-substituted-5-arylidene-thiazolidine-2, 4-dione-isoxazoline derivatives using NaCl/Oxone/Na3PO4 in …

FZ Thari, H Tachallait, NE El Alaoui, A Talha… - Ultrasonics …, 2020 - Elsevier
A rapid and green method for the synthesis of novel N-thiazolidine-2, 4-dione isoxazoline
derivatives 5 from N-allyl-5-arylidenethiazolidine-2, 4-diones 3 as dipolarophiles with …

Synthesis and biological activities of novel chalcone derivatives containing pyrazole oxime ethers

D Hu, N Zhang, Q Zhou, Y Zhou, C Gong, Y Zhang… - Fitoterapia, 2023 - Elsevier
A series of novel chalcone derivatives containing pyrazole oxime ethers were designed and
synthesized. The structures of all the target compounds were determined by NMR and …

Design and Synthesis of C-8 spiro-isoxazoline analogues of 14-Deoxy-11, 12-didehydroandrographolide (14-DDA) for dual targeting of CDK4 and BCL2 mediated …

G Kumar, M Tabassum, BK Sharma, R Kumar… - Journal of Molecular …, 2024 - Elsevier
Deoxy-11, 12-didehydroandrographolide (14-DDA, 3), a secondary metabolite found in
Andrographis paniculata nees, has been synthetically modified into a new series of C-8 …

Ultrasound‐Assisted Green Synthesis of 3,5‐Disubstituted Isoxazole Secondary Sulfonamides via One‐Pot Five‐Component Reaction using CaCl2/K2CO3 as Pre …

AE Mahmoudi, H Tachallait, Z Moutaoukil… - …, 2022 - Wiley Online Library
Tandem one‐pot five‐component reaction involving saccharin, propargyl bromide,
aldehyde, hydroxylamine hydrochloride, and non‐conjugated primary amine has been …

Pharmacophore-based synthesis of pyrazole analogues as artificial antibiotics targeting Salmonella Typhi

H Muniyasamy, MK Aravind, M Arunkumar… - Journal of Molecular …, 2024 - Elsevier
The pharmacological potential of the pyrazole moiety is demonstrated by their presence in a
wide range of therapeutic agents spanning various categories. Notable examples include …

Preparative, mechanistic and tautomeric investigation of 1-phenyl and 1-methyl derivative of 3-methyl-5-pyrazolone

H Fakhraian, Y Nafari - Journal of Chemical Sciences, 2021 - Springer
Phenyl and 1-methyl derivative of 3-methyl-5-pyrazolone were prepared quantitatively via a
scalable solvent-free reaction of corresponding hydrazine derivative with ethyl acetoacetate …

Convenient Synthesis of Pyrazolo[4′,3′:5,6]pyrano[4,3-c][1,2]oxazoles via Intramolecular Nitrile Oxide Cycloaddition

V Milišiūnaitė, E Plytninkienė, R Bakšienė… - Molecules, 2021 - mdpi.com
A simple and efficient synthetic route to the novel 3a, 4-dihydro-3 H, 7 H-and 4 H, 7 H-
pyrazolo [4′, 3′: 5, 6] pyrano [4, 3-c][1, 2] oxazole ring systems from 3-(prop-2-en-1-yloxy) …

A one-pot assembly of Δ2-isoxazolines from ketones, aryl acetylenes and hydroxylamine: Revisiting the mechanism in terms of quantum chemistry

VB Kobychev, AG Pradedova, BA Trofimov - Journal of Molecular Structure, 2021 - Elsevier
A mechanism of the sequential reaction of ketones with arylacetylenes and hydroxylamine in
the presence of KOBu t/DMSO followed by the treatment of the reaction mixture with H 2 O …

Novel aza-bicyclic 2-isoxazoline acylhydrazone hybrids and their synergistic potential with fluconazole against a drug-resistant Candida albicans strain

IKP de Albuquerque, DL de Santana… - Brazilian Journal of …, 2024 - Springer
As the prevalence of drug-resistant Candida isolates continues to rise, the imperative for
identifying novel compounds to enhance the arsenal of antifungal drugs becomes …

[PDF][PDF] Rackauskien e, G.; Arbaciauskien e, E.; Šackus, A. Convenient Synthesis of Pyrazolo [4′, 3′: 5, 6] pyrano [4, 3-c][1, 2] oxazoles via Intramolecular Nitrile …

A Bieliauskas, S Krikštolaityte - Molecules, 2021 - academia.edu
A simple and efficient synthetic route to the novel 3a, 4-dihydro-3H, 7H-and 4H, 7H-pyrazolo
[4′, 3′: 5, 6] pyrano [4, 3-c][1, 2] oxazole ring systems from 3-(prop-2-en-1-yloxy)-or 3 …