Synthesis, antitubercular evaluation and molecular docking studies of phthalimide bearing 1, 2, 3-triazoles

PS Phatak, RD Bakale, ST Dhumal… - Synthetic …, 2019 - Taylor & Francis
In a search for safer and potent antitubercular agents, here a library of newly substituted
dioxoisoindolinylmethyl-triazolyl-N-phenylacetamide derivatives (5a–l) has been …

Identification of 1, 2, 3-triazole-phthalimide derivatives as potential drugs against COVID-19: a virtual screening, docking and molecular dynamic study

VN Holanda, EMA Lima, WV Silva… - Journal of …, 2022 - Taylor & Francis
In this work we aimed to perform an in silico predictive screening, docking and molecular
dynamic study to identify 1, 2, 3-triazole-phthalimide derivatives as drug candidates against …

Synthesis, characterization and cytotoxic activity evaluation of 4-(1, 2, 3-triazol-1-yl) salicylic acid derivatives

ZG Ríos-Malváez, MA Cano-Herrera… - Journal of Molecular …, 2021 - Elsevier
Abstract A novel series of 4-(1, 2, 3-triazol-1-yl) salicylic acid derivatives was synthesized
from 4-azidosalicylic acid and diverse alkynes using copper catalyzed azide-alkyne …

Synthesis and in-vitro biological evaluation of 1, 1-diaryl-2-(1, 2, 3) triazol-1-yl-ethanol derivatives as antifungal compounds flutriafol analogues

JJ García-Vanegas, A Ramírez-Villalva… - Journal of Chemical …, 2019 - Springer
A small library of diverse 1, 1-diaryl-2-(1, 2, 3) triazol-1-yl-ethanol derivatives was designed
and prepared from CuAAC reaction as the key step. The molecular structure of some …

Efficient, mild synthesis of N-unsubstituted 1, 2, 3-triazoles from methanolysis of 1-sulfonyl-1, 2, 3-triazoles

J Rodríguez-Florencio, D Martínez-Otero… - Synthetic …, 2018 - Taylor & Francis
A small library of diverse N-unsubstituted 1, 2, 3-triazoles was prepared from the
corresponding 1-sulfonyl-1, 2, 3-triazoles, which were treated only with MeOH at reflux …

Estudio de la síntesis de 2-alcoxi-N-sulfoniliminas a partir de la inserción de carbenoides derivados de 1-sulfoniltriazoles catalizadas por nanopartículas cobre-hierro

J RODRIGUEZ FLORENCIO - ri.uaemex.mx
La necesidad de proveer nuevas y más eficaces alternativas para el tratamiento
farmacológico de patologías, obliga a las áreas químicas de orgánica, medicinal y …