Transition metal-catalysed cross-coupling is one of the most powerful synthetic methods and
has led to vast improvements in the synthesis of pharmaceuticals, agrochemicals and …

Indole is the most frequently found heterocyclic core structures in pharmaceuticals, natural
products, agrochemicals, dyes and fragrances. For about 150 years, chemists were …

Abstract Unprotected cis‐2, 3‐diarylpiperidines are synthesized through an unprecedented
palladium‐catalyzed cross‐coupling reaction between aryl halides and elusive endocyclic 1 …

An efficient catalytic strategy toward the synthesis of N-substituted 3-methylindoles from
inactive o-dihaloarenes and N-allylamines was developed by using a 1, 3-bis (2, 6 …

An efficient synthesis of N-fused polycyclic indoles by a palladium-catalyzed annulation/acyl
migration cascade reaction is described. The reaction is ligand-free, scalable, and provides …

A practical palladium-catalyzed cascade C–N cross-coupling/Heck reaction of alkenyl
bromides with amino-o-bromopyridines is described for a straightforward synthesis of …

The catalytic deuterodechlorination of aryl/heteroaryl chlorides was developed with a
palladium/unsymmetrical NHC system, and the precisely controlled introduction of …

Background Indoles are important bioactive compounds that have been extensively studied
in organic chemistry. In this work, a green and efficient process for the synthesis of Indoles …

An efficient Mizoroki–Heck/amination cascade reaction of o-dihaloarenes with allylamines
has been developed using nickel and IPr carbene ligand as catalyst. This protocol enables …

A catalytic amount of CuCl and Cs2CO3 was employed to synthesize a variety of 2-
substituted benzo [b] furans and indoles by an intramolecular cyclization of 2-alkynyl …