Catalytic ammoxidation of alcohols into nitriles is an essential reaction in organic synthesis.
While highly desirable, conducting the synthesis at room temperature is challenging, using …

An efficient approach for the construction of enantioenriched γ-azido nitriles through the
chiral sulfide-catalyzed asymmetric electrophilic thioazidation of allylic nitriles is disclosed. A …

The review summarizes and systematizes the literature data on the synthesis and some
aspects of application of pyrrolo [1, 2-a] imidazoles. Synthetic approaches are grouped …

Benzimidazoles, the important scaffold of various biologically important molecules, can be
synthesized using metal catalyzed and metal-free methodologies. Recently, metal-free …

Wittig olefination at hetero-benzylic positions for electron-deficient and electron-rich
heterocycles has been studied. The electronic effects of some commonly used protective …

We report a procedure for the multigram synthesis of 4‐(dimethylamino) pyridinium azide, a
stable, non‐explosive, low‐hygroscopic source of azide ion soluble in both protic and …

A novel approach has been constructed for the synthesis of two types of 2-amino-4-
coumarinyl-5-arylpyrroles (ACAPs, 5 and 6) through a cascade reaction and a metal-free …

To search for potent CDK4/6 covalent inhibitors, total 14 compounds have been designed
and synthesized by connecting different Michael-acceptor to the piperazine moiety of …

The unprecedented synthesis of the indolines bearing N3-quinazolin-2, 4-dione moiety
using an AZIN is reported. The concise synthesis features the tandem Staudinger/chemo …

The kinetics of the ring‐opening reactions of thiophenolates with geminal bis (acceptor)‐
substituted cyclopropanes in DMSO at 20° C was monitored by photometric methods. The …