[PDF][PDF] Synthesis of 1, 3, 4-thiadiazole derivatives and microbiological activities: A review

GAD Barbosa, AP de Aguiar - Rev. Virtual Quim, 2019 - s3.sa-east-1.amazonaws.com
Bacterial resistance associated to different antibiotics is a limitation for the treatment of
infections and this has stimulated the development of new antimicrobial agents. In this …

New 1, 3, 4-thiadiazoles based on thiophene-2-carboxylic acid: Synthesis, characterization, and antimicrobial activities

H Muğlu, H Yakan, HA Shouaib - Journal of molecular structure, 2020 - Elsevier
Abstract Novel 1, 3, 4-thiadiazole derivatives were prepared by cyclization reaction of
thiophene-2-carboxylic acid with N-arylthiosemicarbazides and POCl 3. The antibacterial …

1, 3, 4-Thiadiazole-containing azo dyes: Synthesis, spectroscopic properties and molecular structure

A Kudelko, M Olesiejuk, M Luczynski, M Swiatkowski… - Molecules, 2020 - mdpi.com
Three series of azo dyes derived from 2-amino-5-aryl-1, 3, 4-thiadiazoles and aniline, N, N-
dimethylaniline and phenol were synthesized in high yields by a conventional diazotization …

Straightforward synthesis of 2-chloro-N-(5-(cyanomethyl)-1,3,4-thiadiazol-2-yl)benzamide as a precursor for synthesis of novel heterocyclic compounds with …

AMM Mohamed, MF Ismail, HMF Madkour… - Synthetic …, 2020 - Taylor & Francis
The current work is devoted to the synthesis of 2-chloro-N-(5-(cyanomethyl)-1, 3, 4-
thiadiazol-2-yl) benzamide 5 by an efficient synthetic methodology. The authors decided to …

[HTML][HTML] A combined in vitro and in silico approach of thiadiazole based Schiff base derivatives as multipotent inhibitor: Synthesis, spectral analysis, antidiabetic and …

T Zahoor, S Khan, S Chinnam, T Iqbal, R Hussain… - Results in …, 2024 - Elsevier
We have developed new thiadiazole-containing Schiff base derivatives and examined their
ability to inhibit α-amylase and α-glucosidase. Among the members of series, analogue 1 …

Design, synthesis, and in vitro and in silico studies of 1, 3, 4-thiadiazole-thiazolidinone hybrids as carbonic anhydrase inhibitors

NH Nasab, H Raza, YS Eom, M Hassan… - New Journal of …, 2023 - pubs.rsc.org
In this study, a series of 1, 3, 4-thiadiazole-thiazolidinone derivatives (7a–j) were
synthesized as carbonic anhydrase inhibitors. The in vitro carbonic anhydrase inhibitory …

Synthesis and characterization of 1, 3, 4-thiadiazole compounds derived from 4-phenoxybutyric acid for antimicrobial activities

H Muğlu, N Şener, HAM Emsaed, S Özkınalı… - Journal of Molecular …, 2018 - Elsevier
Abstract New 1, 3, 4-thiadiazole compounds were synthesized through the cyclization
reaction of 4-phenoxybutyric acid and N-phenylthiosemicarbazide derivatives with …

Synthesis, dyeing performance and evaluation of the antimicrobial and antioxidant activities of azo dye derivatives incorporated with 1, 3, 4-thiadiazole combined with …

K Mezgebe, Y Melaku, VP Ramachandran… - New Journal of …, 2024 - pubs.rsc.org
The incorporation of heterocyclic moieties into azo dye derivatives influences the bioactive
properties of synthesized derivatives. Herein, six azo dye derivatives incorporated with 1, 3 …

Design, synthesis, and characterization of a novel pH-responsive azo dye incorporating a 1, 3, 4-thiadiazole ring for advanced textile applications

S Belowar, M Rahamatolla, S Islam, MA Jalil… - Dyes and …, 2024 - Elsevier
This study presents the synthesis and comprehensive characterization of a novel azo dye
derived from 2-(5-amino-1, 3, 4-thiadiazol-2-yl) phenol (1a). The synthesis was initiated by …

Synthesis, Characterization, and Antimicrobial Properties of New 1, 3, 4‐Thiadiazoles Derived from Azo Dyes

M Gür - Journal of Heterocyclic chemistry, 2019 - Wiley Online Library
Some new 1, 3, 4‐thiadiazoles derived from azo dyes were synthesized. Two different
synthesis methods were used for these compounds: Esters pertaining to the azo dyes were …