Investigation and comparison of biological effects of regioselectively synthesized thiazole derivatives

M Moghaddam‐manesh, H Beyzaei… - Journal of …, 2021 - Wiley Online Library
In this study, anticancer, antibacterial (against hospital‐isolated antibiotic‐resistant
Escherichia coli strains), antifungal, and antioxidant effects of synthesized heterocyclic …

Synthesis, characterization and in-vitro anti-inflammatory activity of some substituted 1, 2, 3, 4 tetrahydropyrimidine derivatives

AS Gondkar, VK Deshmukh, SR Chaudhari - Drug Invention Today, 2013 - Elsevier
Background & aim Pyrimidines represent a broad class of compounds, which have received
considerable attention due to their wide range of biological activities such as, anti …

Synthesis, in vitro and in silico studies of novel potent urease inhibitors: N-[4-({5-[(3-Un/substituted-anilino-3-oxopropyl) sulfanyl]-1, 3, 4-oxadiazol-2-yl} methyl)-1, 3 …

MA Abbasi, M Hassan, SZ Siddiqui, H Raza… - Bioorganic & medicinal …, 2018 - Elsevier
The present article describes the synthesis, in vitro urease inhibition and in silico molecular
docking studies of a novel series of bi-heterocyclic bi-amides. The synthesis of title …

A comparative study on the antibacterial effects of some newly synthesized thiazole, imidazolidine and tetrahydropyrimidine derivatives against Bacillus cereus and …

B Ghasemi, H Beyzaie, H Majidiani - Pharmaceutical Sciences, 2016 - ps.tbzmed.ac.ir
Background: Bacillus cereus and Salmonella typhimurium are important human pathogenic
bacteria. The spread of strains of drug-resistant these pathogens has encouraged …

Regioselective synthesis of 2-[(E)-(benzo[d]thiazol-2(3H)-ylidene)(cyano)methyl]thiazoles

M Bakavoli, H Beyzaei, M Rahimizadeh, H Eshghi - 2011 - degruyter.com
Abstract Cyclocondensation of 2-[bis (methylthio) methylene] malononitrile and 2-amino-
benzenthiol afforded 2-(benzo [d] thiazol-2-yl) malononitrile. This compound, on treatment …

[PDF][PDF] Evaluation of antibacterial effects of benzothiazole derivatives on bacterial food pathogens

B Ghasemi - Iran J Med Microbiol: Volume, 2015 - ijmm.ir
Materials and Methods: Synthesized thiazole derivatives were prepared in DMSO. Well
method was used for the calculation of growth inhibition zone diameters and serial dilution …

[PDF][PDF] Synthesis of some derivatives of 4-phenyl-1, 3-dihydro-2H-imidazole-2-thion using ionic liquid as catalyst and evaluation of their antimicrobial activity

U Onn - International Journal of Chemistry, 2017 - pdfs.semanticscholar.org
Abstract The synthesis of some 1, 3-diazoles and thiazoles was realized in different
conditions: a) In the presence of PTSA or sulfuric acid as catalyst we obtained only diazole …

Study of antibacterial effect of novel thiazole, imidazole, and tetrahydropyrimidine derivatives against Listeria monocytogenes

B Ghasemi, H Beyzaei, H Hashemi - Annals of Military and Health …, 2015 - brieflands.com
: Purpose: In this study, we have focused on antibacterial effect of newly synthesized
thiazole, imidazole, and tetrahydropyrimidine derivatives in Iran on listeria monocytogenes …

Study of antibacterial effect of new thiazole, thiazolidine, imidazole, tetrahydropyrimidine, oxazolidine and thiazepine derivatives against Enterococcus faecalis

H Beyzaei, MR Moghadam Manesh - Yafte, 2016 - eprints.lums.ac.ir
Background: To resistant of Enterococcus faecalis to a range of antibiotics, has become one
of the concerns of sanitation in most communities and has made many researchers raise …

Reactions of ketene dithioacetal for a new versatile synthesis of 4, 5-substituted 3-aminothiophene-2-carboxylate derivatives

SM Chavan, RB Toche, VM Patil… - Journal of Sulfur …, 2016 - Taylor & Francis
Poly substituted 3-aminothiophenes were successfully synthesized in good yields by using a
one-pot protocol via ketene S, S-acetal as an intermediate in basic medium (K2CO3/N, N …