Cell cycle inhibition, apoptosis, and molecular docking studies of the novel anticancer bioactive 1, 2, 4-triazole derivatives

J Ghanaat, MA Khalilzadeh, D Zareyee… - Structural Chemistry, 2020 - Springer
Abstract Several 3-alkylsulfanyl-1, 2, 4-triazole derivatives were synthesized and their
relevant structures confirmed based on their elemental analysis and nuclear magnetic …

Stereoselective synthesis of dihydrothiadiazinoazines and dihydrothiadiazinoazoles and their pyrolytic desulfurization ring contraction

A Al-Etaibi, E John, MR Ibrahim, NA Al-Awadi… - Tetrahedron, 2011 - Elsevier
Intramolecular base catalyzed C–C bond formation led to exclusive stereoselective
syntheses of trans-6, 7-dihydro-5H-[1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazines, trans-7, 8 …

Synthesis of spiro derivatives of 1,2,3-triazolo[5,1-b][1,3,4]thiadiazines and biological activity thereof

TA Kalinina, OA Bystrykh, VA Pozdina… - Chemistry of …, 2015 - Springer
3-Cyclopentylidene (cyclohexylidene) amino-3 H-1, 2, 3-triazole-4-thiolates, formed via
Dimroth rearrangement of 1, 2, 3-thiadiazolylhydrazones of cyclopentanone and …

Intramolecular Cyclization of the ortho‐Substituted N‐arylquinone Imines under Basic and Thermal Conditions

ES Khodykina, DV Steglenko, EV Vetrova… - …, 2023 - Wiley Online Library
Abstract The S (O, N)‐benzyl ethers of N‐arylquinone imines undergo cyclization under the
action of bases to form products of the benzothiazol, benzoxazole, and benzimidazole …

6,7‐Dihydro‐5H‐1,2,4‐triazolo[3,4‐b][1,3,4]thiadiazine Ring Cleavage and Tautomerism of the Products: Experimental and Theoretical Study

AA Kolodina, AA Tsaturyan, MS Galkina… - …, 2020 - Wiley Online Library
Electronic effects of aryl substituents at the C (7)‐atom play a crucial role in the cleavage of a
six‐membered ring of 6, 7‐dihydro‐5H‐[1, 2, 4] triazolo [3, 4‐b][1, 3, 4] thiadiazines. Our …

Recent progress in the synthetic routes to triazolothiadiazines

BF Abdel-Wahab, I Althagafi - … , Sulfur, and Silicon and the Related …, 2014 - Taylor & Francis
Full article: Recent Progress in the Synthetic Routes to Triazolothiadiazines Skip to Main
Content Taylor and Francis Online homepage Taylor and Francis Online homepage Log in …

Unusual cyclization of N-imidazolyl quinone imines with the formation of thiadiazole ring and its subsequent recyclization

AA Kolodina, DV Steglenko, ES Khodykina… - Mendeleev …, 2022 - Elsevier
Di-tert-butyl-4-{[2-(2-aryl-2-oxoethylthio)-1H-imidazol-1-yl] imino} cyclohexa-2, 5-dien-1-
ones under the action of bases give products of the 2, 3-dihydroimidazo [2, 1-b] thiazol-3-ol …

CИНТЕЗ И БИОЛОГИЧЕСКАЯ АКТИВНОСТЬ СПИРОПРОИЗВОДНЫХ 1,2,3-ТРИАЗОЛО[5,1-b][1,3,4]ТИАДИАЗИНОВ

ТА Калинина, ОA Быстрых, ВА Поздина… - Chemistry of …, 2015 - osi131.osi.lv
Перегруппировкой Димрота 1, 2, 3-тиадиазолилгидразонов циклопентанона и
циклогексанона в присутствии триэтиламина были получены 3-циклопентилиден …

Synthesis and crystal structure of ((6R,7S)-3-ethyl-6-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl)(phenyl)methanone hemihydrate, 2(C19H18N4OS) ⋅ H …

Q Ding, R Yang, P Yao - Zeitschrift für Kristallographie-New Crystal …, 2020 - degruyter.com
Synthesis and crystal structure of ((6R,7S)-3-ethyl-6-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl)(phenyl)methanone
hemihydrate, 2(C19H18N4OS) ⋅ H2O Skip to content Should you have institutional access …

Bazı yeni kondanse triazol türevlerinin sentezi ve antikanser aktivitelerinin araştırılması

SP Aytaç - 2015 - acikbilim.yok.gov.tr
Bu çalışmada antikanser etki göstermesi beklenen, 4-amino-3-sübstitüe-1, 2, 4-triazol-5-
tiyon (Bileşik 1-3), 3, 6-disübstitüe-7H-1, 2, 4-triazolo [3, 4-b]-1, 3, 4-tiyadiazin (Bileşik 1a-3j) …