M Luczynski, A Kudelko - Applied Sciences, 2022 - mdpi.com
Biologically active compounds play a key role in the fight against diseases affecting both human and animal living organisms, as well as plants. Finding out about new molecules …
Current study is based on the sequential conversion of indolyl butanoic acid (1) into ethyl indolyl butanoate (2), indolyl butanohydrazide (3), and 1, 3, 4-oxadiazole-2-thiol analogs (4) …
This study reports the synthesis, biological investigation and molecular docking of novel β- lactam derivatives bearing 1, 3, 4-thiadiazole and 1, 3, 4-oxadiazole ring system. The …
In the study presented herein, 4-(1H-indol-3-yl) butanoic acid (1) was sequentially transformed in the first phase into ethyl 4-(1H-indol-3-yl) butanoate (2), 4-(1H-indol-3-yl) …
MB Taj, A Raheel, W Alelwani, N Babteen… - Russian Journal of …, 2019 - Springer
Abstract Ten N (N′)-arylbenzamidines were synthesized in 60–77% yield by one-pot microwave-assisted reaction of the corresponding N-arylbenzamides with aniline or …
MNAM Taib, NS Hasmaruddin, NAM Ali, H Osman… - 2022 - researchsquare.com
Abstract A series of new 2, 5-disubstituted-1, 3, 4-oxadiazole derivatives (5a-j and 6a-j) have been designed and synthesized in four-steps. sixteen compounds among the twenty …
Abstract Background: 1, 3, 4-Oxadiazole have been reported for the diverse use in medicine because of its versatile pharmacological properties. In continuation of our on-going research …
In the study presented here, the nucleophilic substitution reaction of 5-[3-(1H-indol-3-yl) propyl]-1, 3, 4-oxadiazol-2-ylhydrosulfide was carried out with different alkyl/aralkyl halides …
MNA Mohamad Taib, NS Hasmaruddin… - Zaheen and Abd Ghani … - papers.ssrn.com
A series of new 2-alkylbenzysulfanyl-5-substituted-1, 3, 4-oxadiazoles derivatives (5a-j and 6a-j) were synthesized in four-step reaction from carboxylic acid analogues as the starting …