Application of the Suzuki-Miyaura reaction in the synthesis of flavonoids
MA Selepe, FR Van Heerden - Molecules, 2013 - mdpi.com
The application of the Suzuki-Miyaura reaction in the synthesis of flavonoids, an important
class of natural products, is reviewed. This reaction has not only been employed to provide …
class of natural products, is reviewed. This reaction has not only been employed to provide …
Stereoselective synthesis of flavonoids: A brief overview
AM Pereira, H Cidade, ME Tiritan - Molecules, 2023 - mdpi.com
Stereoselective synthesis has been emerging as a resourceful tool because it enables the
obtaining of compounds with biological interest and high enantiomeric purity. Flavonoids are …
obtaining of compounds with biological interest and high enantiomeric purity. Flavonoids are …
Los compuestos fenólicos, un acercamiento a su biosíntesis, síntesis y actividad biológica
DAM Gordo - RIAA, 2018 - dialnet.unirioja.es
Los compuestos fenólicos hacen parte de uno de los grupos más abundantes dentro de los
metabolitos secundarios. Éstos se biosintetizan en las plantas por medio de rutas como la …
metabolitos secundarios. Éstos se biosintetizan en las plantas por medio de rutas como la …
A facile route to flavone and neoflavone backbones via a regioselective palladium catalyzed oxidative Heck reaction
A straightforward and atom-economical base-free palladium-catalyzed regioselective direct
arylation of coumarins and chromenones is devised. This protocol is compatible with a wide …
arylation of coumarins and chromenones is devised. This protocol is compatible with a wide …
Simple coumarins: privileged scaffolds in medicinal chemistry
MFM Borges, FMF Roleira… - … Chemistry: Volume 4, 2009 - benthamdirect.com
Coumarins, also known as benzopyrones, are present in remarkable amounts in plants,
although their presence has also been detected in microorganisms and animal sources. The …
although their presence has also been detected in microorganisms and animal sources. The …
Palladium-catalyzed oxidative Heck coupling reaction for direct synthesis of 4-arylcoumarins using coumarins and arylboronic acids
An efficient protocol for the direct synthesis of 4-arylcoumarins via palladium-catalyzed
oxidative Heck coupling reaction of coumarins and arylboronic acids was developed. 4 …
oxidative Heck coupling reaction of coumarins and arylboronic acids was developed. 4 …
Photoinduced generation of acyl radicals from simple aldehydes, access to 3-acyl-4-arylcoumarin derivatives, and evaluation of their antiandrogenic activities
K Kawaai, T Yamaguchi, E Yamaguchi… - The Journal of …, 2018 - ACS Publications
A novel photocatalysis to construct the 3-acyl-4-arylcoumarin framework from simple
aldehyde with ynoate is described. The reaction proceeded through an acyl radical …
aldehyde with ynoate is described. The reaction proceeded through an acyl radical …
[HTML][HTML] SLC26A3 inhibitor identified in small molecule screen blocks colonic fluid absorption and reduces constipation
SLC26A3 (downregulated in adenoma; DRA) is a Cl–/anion exchanger expressed in the
luminal membrane of intestinal epithelial cells, where it facilitates electroneutral NaCl …
luminal membrane of intestinal epithelial cells, where it facilitates electroneutral NaCl …
Syntheses and biological activities of chroman-2-ones. A review
Chroman-2-one (1), also referred to as dihydrocoumarin, and its derivatives have attracted
the attention of chemists due to their broad range of properties. Dihydrocoumarin contains a …
the attention of chemists due to their broad range of properties. Dihydrocoumarin contains a …
Recent advances in transition-metal-catalyzed synthesis of coumarins
Coumarin is a privileged scaffold found in a large number of biologically active natural
products, pharmaceuticals and agrochemicals, and functionalized coumarins are also …
products, pharmaceuticals and agrochemicals, and functionalized coumarins are also …