[HTML][HTML] The Molecular Architecture of Pseudomonas aeruginosa Quorum-Sensing Inhibitors

Q Li, S Mao, H Wang, X Ye - Marine Drugs, 2022 - mdpi.com
The survival selection pressure caused by antibiotic-mediated bactericidal and bacteriostatic
activity is one of the important inducements for bacteria to develop drug resistance. Bacteria …

[HTML][HTML] Small Schiff Base Molecules—A Possible Strategy to Combat Biofilm-Related Infections

M Coandă, C Limban, DC Nuță - Antibiotics, 2024 - mdpi.com
Microorganisms participating in the development of biofilms exhibit heightened resistance to
antibiotic treatment, therefore infections involving biofilms have become a problem in recent …

[HTML][HTML] Screening of natural product derivatives identifies two structurally related flavonoids as potent quorum sensing inhibitors against gram-negative bacteria

S Manner, A Fallarero - International journal of molecular sciences, 2018 - mdpi.com
Owing to the failure of conventional antibiotics in biofilm control, alternative approaches are
urgently needed. Inhibition of quorum sensing (QS) represents an attractive target since it is …

[HTML][HTML] Physicochemical studies on the inhibitive properties of a 1, 2, 4-triazole Schiff's base, HMATD, on the corrosion of mild steel in hydrochloric acid

PR Ammal, M Prajila, A Joseph - Egyptian Journal of Petroleum, 2018 - Elsevier
Abstract The efficiency of 4-(4-hydroxy-3-methoxy benzyledene amino)-4-H-1, 2, 4-triazole-
3, 5-dimethanol, HMATD, as corrosion inhibitor for mild steel in 0.5 M HCl has been …

Microwave assisted green synthesis, Single crystal XRD, DFT, Hirshfeld surface analysis, Antibiofilm, Anti-inflammatory activity and Molecular docking study of 4-(4 …

D Bhosale, A Narale, D Raut, M Bamankar… - Journal of Molecular …, 2023 - Elsevier
Abstract The title compound 4-(4-Fluorophenyl)-5-methyl-1, 3-thiazole-2-amine was
synthesized by the green microwave irradiation method and the structure was confirmed by …

Novel Schiff base derivatives containing 4, 5-disubstituted thiazole as potential antibiofilm, anti-inflammatory and antioxidant agents: Green synthesis, molecular …

D Bhosale, A Narale, P Hadimani, M Kokane… - Journal of Molecular …, 2024 - Elsevier
We report the microwave-assisted (MW) green synthesis of some novel 4, 5 disubstituted
thiazole-containing Schiff base derivatives (SBs) as antibiofilm, anti-inflammatory, and …

Synthesis and anti-biofilm activity of thiazole Schiff bases

PG More, NN Karale, AS Lawand, N Narang… - Medicinal Chemistry …, 2014 - Springer
A series of thiazole Schiff bases (SB-1 to SB-7) have been synthesized by reacting 4-(o-
methoxyphenyl)-2-aminothiazole and R substituted salicylaldehyde (R= H, 3-Me, 4-Me, 5 …

NBS-mediated sequential one-pot synthesis of multifunctionalized thiazoles and thiophenes from 1, 3-dicarbonyl compounds and mercaptonitrile salts

L Luo, L Meng, Q Sun, Z Ge, R Li - Tetrahedron Letters, 2014 - Elsevier
A NBS-mediated sequential one-pot synthesis of multifunctionalized thiazoles and
thiophenes from 1, 3-dicarbonyl compounds and mercaptonitrile salts has been developed …

[PDF][PDF] Anti-quorum sensing activity of 1, 3-dihydro-2H-benzimidazol-2-one derivatives

E Onem, Y Dundar, S Ulusoy, N Noyanalpan… - Fresenius Environ …, 2018 - researchgate.net
Many Gram-negative bacteria use N-acyl homoserine lactone (AHL) signal molecules to
monitor their own population density and coordinate gene regulation in a process called …

[PDF][PDF] The Importance of 2-AminoThiazole Schiff Bases as Antimicrobial and Anticancer Agents.

SL Abdulhadi, MQ Abdulkadir… - Al-Mustansiriyah Journal of …, 2020 - iasj.net
The pharmacophore 2-aminothiazole has an interesting role in pharmaceutical chemistry as
this led to the synthesis of many types of compounds with diverse biological activity. Schiff …