A newly series of 4-(phenylurenyl) chalcone (4a–j) and 4′-(phenylurenyl/thiourenyl)
chalcone (9a–l) derivatives were synthesized and their inhibitory effects on the diphenolase …

A novel series of donepezil-trolox hybrids were designed, synthesized, and evaluated as
multifunctional ligands against Alzheimer's disease (AD). Biological assays showed that …

A newly series of 6-(phenylurenyl/thiourenyl) saccharin (6a–y) derivatives were synthesized
and their inhibitory effects on the diphenolase activity of banana tyrosinase were evaluated …

A new series of 1, 3, 4-oxadiazole-3 (2H)-carboxamide derivatives have been synthesized
by direct heterocyclization reaction of substituted benzoylisocyanate with various …

Two series of 1, 3, 4-oxadiazoline heterocycle derivatives were designed, synthesized and
identified. Bioactivity assays showed that all synthesized compounds inhibited chitin …

Abstract In this study, 4'-(phenylurenyl/thiourenyl) chalcones (14–25) were prepared from 4'-
(phenylurenyl/thiourenyl) acetophenones and benzaldehyde derivatives by Claisen-Schmidt …

A facile synthetic approach towards dithiatetraaza-macrocycles 4a and b was achieved
through reaction of 2, 2′-[alkanediylbis (thio)] bisbenzenamines 1a and b with 1, 4 …

Ever since the idea arose that melatonin might promote sleep and resynchronize circadian
rhythms, many research groups have centered their efforts on obtaining new melatonin …

The goal of this study was the design and synthesis of bulky and polar-bulky
galactonoamidines that have a potential to interact with both catalytic amino acids in the …

Melanin-concentrating hormone (MCH) regulates feeding and energy homeostasis through
interaction with its receptor, the melanin-concentrating receptor 1 (MCHR1), making it a …