[HTML][HTML] The Synthesis and Evaluation of Aminocoumarin Peptidomimetics as Cytotoxic Agents on Model Bacterial E. coli Strains

P Kowalczyk, M Wilk, P Parul, M Szymczak… - Materials, 2021 - mdpi.com
This work presents the successful synthesis of a library of novel peptidomimetics via Ugi
multicomponent reaction. Most of these peptidomimetics contain differently substituted …

Synthesis and characterization of bis-amide SSE1917 as a microtubule-stabilizing anticancer agent

S Iqbal, F Firdous, M Furqan, A Bilal, S Fozail… - Bioorganic …, 2024 - Elsevier
Microtubule dynamics are critical for spindle assembly and chromosome segregation during
cell division. Pharmacological inhibition of microtubule dynamics in cells causes prolonged …

[HTML][HTML] Garlic extract: inhibition of biochemical and biophysical changes in glycated HSA

MWA Khan, AA Otaibi, AFM Alhumaid, AKD Alsukaibi… - Applied Sciences, 2021 - mdpi.com
Glycation of various biomolecules contributes to structural changes and formation of several
high molecular weight fluorescent and non-fluorescent, advanced glycation end products …

Unveiling the versatility of novel oxacalix [4] arene platform: Systematic screening and comparative study on biological and antioxidant potency

BK Seth, S Dey, P Trivedi, G Sindhav… - Journal of Molecular …, 2024 - Elsevier
Calixarene, a third generation supramolecule, have made their signature in biomedical
applications through their unique physicochemical characteristics. Oxacalixarene, a class of …

[PDF][PDF] The Synthesis of Aminocoumarin Peptidomimetics and Evaluation as a Cytotoxic on Model Bacterial E. coli Strains. Materials 2021, 14, 5725

P Kowalczyk, M Wilk, P Sahrawat, M Szymczak… - 2021 - academia.edu
This work presents the successful synthesis of a library of novel peptidomimetics via Ugi
multicomponent reaction. Most of these peptidomimetics contain differently substituted …