As one of the most important structural units in pharmaceuticals and medicinal chemistry,
quinazolinone and its derivatives exhibit a wide range of biological and pharmacological …

Herein, a metal-and photosensitizer-free protocol has been developed for decarboxylative C–
H (amino) alkylation of heteroarenes using carboxylic acids as the (amino) alkylating …

Utilization of oxime esters as bifunctional reagents in energy-transfer photocatalysis has
received considerable attention. However, the reaction type is so far limited to the …

Although photocatalytic C− H activation has been realized by using heterogeneous
catalysts, most of them require high‐temperature conditions to provide the energy required …

The pyridine core is a crucial component in numerous FDA‐approved drugs and
Environmental Protection Agency (EPA) regulated agrochemicals. It also plays a significant …

The development of ligands and the elucidation of their roles in the catalytic cycle are key to
achieving high efficiency and selectivity in nondirected transition-metal-catalyzed C–H …

Molecular editing promises to facilitate the rapid diversification of complex molecular
architectures by rapidly and conveniently altering core frameworks. This approach has the …

Herein, we report a protocol for the stereoselective C–H alkenylation of five-membered
heteroarenes including pyrroles (containing free NH pyrrole), thiophenes, and furans with 1 …

Herein, we report that the dipole moments of tautomers can be the controlling factor for
regiodivergent synthesis of either 14 H-quinazolino [3, 2-f] phenanthridin-14-ones or 6 H …

An efficient PdII-and RhIII-controlled site-selective C–H bond alkynylation of
imidazopyridines using (bromoethynyl) triisopropylsilane is disclosed. The divergent …