Repositioning of acefylline as anti-cancer drug: Synthesis, anticancer and computational studies of azomethines derived from acefylline tethered 4-amino-3-mercapto …
Novel azomethines derived from acefylline tethered triazole hybrids (7a-k) have been
synthesized and evaluated against human liver cancer cell line (Hep G2) using MTT assay …
synthesized and evaluated against human liver cancer cell line (Hep G2) using MTT assay …
Unfolding the antibacterial activity and acetylcholinesterase inhibition potential of benzofuran-triazole hybrids: Synthesis, antibacterial, acetylcholinesterase inhibition …
In this study, a series of novel benzofuran-based 1, 2, 4-triazole derivatives (10a–e) were
synthesized and evaluated for their inhibitory potential against acetylcholinesterase (AChE) …
synthesized and evaluated for their inhibitory potential against acetylcholinesterase (AChE) …
In-vitro cytotoxic evaluation of newly designed ciprofloxacinoxadiazole hybrids against human liver tumor cell line (Huh7).
Fluoroquinolones are targets of interest due to their broad spectrum antibacterial activity.
Structure-activity relationship (SAR) of fluoroquinolones clearly indicates that substitution at …
Structure-activity relationship (SAR) of fluoroquinolones clearly indicates that substitution at …
Ultrasound-assisted synthesis and in silico modeling of methanesulfonyl-piperazine-based dithiocarbamates as potential anticancer, thrombolytic, and hemolytic …
Piperazine-based dithiocarbamates serve as important scaffolds for numerous
pharmacologically active drugs. The current study investigates the design and synthesis of a …
pharmacologically active drugs. The current study investigates the design and synthesis of a …
Facile green approach towards the synthesis of some phenyl piperazine based dithiocarbamates as potent hemolytic and thrombolytic agents.
The facile and efficient protocol for the synthesis of N-phenyl piperazine based di-thio-
carbamates has been reported under neat conditions. A library of novel piperazine based di …
carbamates has been reported under neat conditions. A library of novel piperazine based di …
Facile one-pot approach to the synthesis of alkyl piperazine-1-carbodithioates as hemolytic and thrombolytic agents
A polyethylene glycol (PEG)-promoted methodology has been utilized for synthesis of
piperazine-based dithiocarbamates. One-pot reaction of N-methylpiperazine and N-Boc …
piperazine-based dithiocarbamates. One-pot reaction of N-methylpiperazine and N-Boc …
[PDF][PDF] Facile synthesis, antibacterial and protease inhibition studies of β-amino alcohols prepared via ring opening of epoxides.
A green ultrasound assisted convenient approach has been reported for the ring opening of
epoxides. As a result, a series of N-phenyl piperazine and morpholine based β-amino …
epoxides. As a result, a series of N-phenyl piperazine and morpholine based β-amino …
2-{[4-(4-Bromophenyl)piperazin-1-yl)]methyl}-4-(3-chlorophenyl)-5-(4-methoxyphenyl)-2,4-dihydro-3H-1,2,4-triazole-3-thione
M Wujec, R Typek - Molbank, 2023 - mdpi.com
The novel compound 2-{[4-(4-bromophenyl) piperazin-1-yl)] methyl}-4-(3-chlorophenyl-5-(4-
methoxyphenyl)-2, 4-dihydro-3 H-1, 2, 4-triazole-3-thione is obtained in good yield via a …
methoxyphenyl)-2, 4-dihydro-3 H-1, 2, 4-triazole-3-thione is obtained in good yield via a …
[PDF][PDF] triazole-3-thione
M Wujec, R Typek - 2023 - ppm.umlub.pl
Piperazine is a common structural motif found in agrochemicals and pharmaceuticals, in part
due to its ability to positively modulate the pharmacokinetic properties of a drug substance …
due to its ability to positively modulate the pharmacokinetic properties of a drug substance …
[PDF][PDF] Repositioning of acefylline as anti-cancer drug: Synthesis, anticancer and computational studies of azomethines derived from acefylline tethered 4-amino-3 …
N Anjum, AIID Azhar Rasul, K Kotwica-Mojzych - ppm.umlub.pl
Novel azomethines derived from acefylline tethered triazole hybrids (7a-k) have been
synthesized and evaluated against human liver cancer cell line (Hep G2) using MTT assay …
synthesized and evaluated against human liver cancer cell line (Hep G2) using MTT assay …