1, 1, 1, 3, 3, 3-Hexafluoroisopropanol (HFIP) is a polar, strongly hydrogen bond-donating
solvent that has found numerous uses in organic synthesis due to its ability to stabilize ionic …

The reactivity and selectivity of 1, 3‐diynes in transition‐metal‐catalyzed C H activation is
exploited to quickly assemble diverse polysubstituted bisheterocycles, which are highly …

In this paper, a highly efficient and regioselective synthesis of pyrazolone fused
benzodiazepine derivatives via the reaction of 1-phenylpyrazolidinones with propargyl …

An unprecedented divergent synthesis of pyrazolo [1, 2-a] pyrazolones and 2-acylindoles
via Rh (III)-catalyzed [4+ 1] or [3+ 2] annulation of 1-phenylpyrazolidinones with alkynyl …

Herein, a novel synthesis of pyrazolidinone fused 1, 3-benzooxazepine derivatives via a
formal [4+ 3] annulation reaction of 1-phenylpyrazolidinones with diazonaphthalen-2 (1H) …

The ability to establish switchable site-selectivity through catalyst control in the direct
functionalization of molecules that contain distinct C–H bonds remains a demanding …

Here a new, mild and versatile method for one-pot cascade synthesis of diverse N-
methoxyisoquinolinediones via Rh (III)-catalyzed regioselective carbenoid insertion C–H …

A highly efficient iridium-catalyzed cascade annulation of pyrazolones and sulfoxonium
ylides to access various pyrazolo [1, 2-α] cinnoline derivatives has been achieved. This …

A rhodium (III)-catalyzed controllable [4+ 1] and [4+ 2] annulation of N-aryl pyrazolones with
maleimides as C1 and C2 synthon has been explored for the synthesis of spiro [pyrazolo [1 …

Presented herein is a controllable selective construction of spiro or fused heterocyclic
scaffolds through the one-pot cascade reactions of 1-phenylpyrazolidinones with …