Preparation of shell-core fiber-encapsulated Lactobacillus rhamnosus 1.0320 using coaxial electrospinning

C Xu, J Ma, Z Liu, W Wang, X Liu, S Qian, L Chen, L Gu… - Food Chemistry, 2023 - Elsevier
In this study, shell-core fibers were successfully prepared by using Eudragit S100 (ES100)
and poly (vinyl alcohol)(PVA)/pectin (PEC) through coaxial electrospinning technology. The …

Synthesis and molecular docking of some novel 3-thiazolyl-coumarins as inhibitors of VEGFR-2 kinase

TZ Abolibda, M Fathalla, B Farag, MEA Zaki… - Molecules, 2023 - mdpi.com
One crucial strategy for the treatment of breast cancer involves focusing on the Vascular
Endothelial Growth Factor Receptor (VEGFR-2) signaling system. Consequently, the …

Design, synthesis, anticancer activity and docking studies of novel quinazoline-based thiazole derivatives as EGFR kinase inhibitors

MS Raghu, HA Swarup, T Shamala, BS Prathibha… - Heliyon, 2023 - cell.com
The in vitro anticancer efficacy of a new series of quinazoline-based thiazole derivatives was
explored. Three cancer cell lines, MCF-7, HepG2, and A548, as well as the normal Vero cell …

Pt (IV) and Au (III) complexes with tridentate-benzothiazole based ligand: Synthesis, characterization, biological applications (antibacterial, antifungal, antioxidant …

HAK Kyhoiesh, KJ Al-Adilee - Inorganica Chimica Acta, 2023 - Elsevier
A novel tridentate azo dye ligand, 2-[2′-(6-methoxybenzothiazolyl) azo]-5-dimethylamino
benzoic acid (6-MBTADB) and its Pt (IV) and Au (III) metal complexes have been …

Synthesis, in-vitro α-glucosidase inhibition and molecular docking studies of 1, 3, 4-thiadiazole-5, 6-diphenyl-1, 2, 4-triazine hybrids: potential leads in the search of …

H Kumar, M Dhameja, S Kurella, A Uma… - Journal of Molecular …, 2023 - Elsevier
Abstract A series of 1, 3, 4-thiadiazole-5, 6-diphenyl-triazine hybrids 7a-l have been
designed, synthesized and investigated for the α-glucosidase inhibitory activities. All the …

In-situ coordination assembly of polyphenol with cage-like Prussian blue as an ecofriendly nanocarrier for site-specific pesticide delivery and sustained pest control

L Zhang, M Fang, C Yang, F Zhang, Z Lu… - Journal of Cleaner …, 2024 - Elsevier
In sustainable agricultural production, an efficient and environmental-friendly nanoplatform
for precise pesticide delivery is considerably desirable to enhance efficacy and minimize …

Design and synthesis of novel benzimidazole linked thiazole derivatives as promising inhibitors of drug-resistant tuberculosis

K Veena, MS Raghu, KY Kumar, CBP Kumar… - Journal of Molecular …, 2022 - Elsevier
Despite combination therapy is effective in treating tuberculosis (TB) caused by susceptible
Mycobacterium tuberculosis (Mtb) strains, overcoming multidrug resistance (MDR) remains …

Synthesis and biological activity, and molecular modelling studies of potent cytotoxic podophyllotoxin-naphthoquinone compounds

HT Nguyen, QGN Thi, THN Thi, PH Thi… - RSC …, 2022 - pubs.rsc.org
A new approach for the synthesis of podophyllotoxin-naphthoquinone compounds using
microwave-assisted three-component reactions is reported in this study. Novel …

[HTML][HTML] Impact of polar (DMSO, ethanol, water) solvation on geometry, spectroscopy (FT-IR, UV, NMR), quantum chemical parameters, and the antifungal activities of …

OC Godfrey, I Anna, SW Qader, G Sampathkumar… - Chemical Physics …, 2023 - Elsevier
Due to their ubiquity and the rise of drug-resistant forms, Candida albicans infections pose a
serious threat to world health. Exploring new molecular possibilities is essential in order to …

Design, synthesis and molecular docking studies of imidazole and benzimidazole linked ethionamide derivatives as inhibitors of InhA and antituberculosis agents

MS Raghu, CBP Kumar, KY Kumar… - Bioorganic & Medicinal …, 2022 - Elsevier
To explore effective antituberculosis agents, a new class of imidazoles and benzimidazoles
linked ethionamide analogs were designed and synthesized. The elemental analysis, 1 H …