The conjugate addition of enantiomerically pure lithium amides as homochiral ammonia equivalents: scope, limitations and synthetic applications

SG Davies, AD Smith, PD Price - Tetrahedron: Asymmetry, 2005 - Elsevier
The conjugate addition of enantiomerically pure lithium amides as homochiral ammonia
equivalents: scope, limitations and synthetic applications - ScienceDirect Skip to main contentSkip …

Direct-type catalytic three-component mannich reactions leading to an efficient synthesis of α, β-diamino acid derivatives

MM Salter, J Kobayashi, Y Shimizu, S Kobayashi - Organic Letters, 2006 - ACS Publications
The first example of the Lewis acid-catalyzed three-component direct-type Mannich reaction
of simple aromatic and enolizable aliphatic aldehydes, secondary amines, and glycine …

An Efficient Synthesis of 2- and 2,6-Substituted Piperidines Using PdII-Catalyzed 1,3-Chirality Transfer Reaction

SM Hande, N Kawai, J Uenishi - The Journal of Organic …, 2009 - ACS Publications
An efficient and general method for 2-and 2, 6-substituted piperidine syntheses using PdII-
catalyzed 1, 3-chirality transfer reaction has been developed. The various N-protected ζ …

Access to 2, 6-disubstituted piperidines: control of the diastereoselectivity, scope, and limitations. applications to the stereoselective synthesis of (−)-solenopsine A and …

I Abrunhosa-Thomas, A Plas, A Vogrig… - The Journal of …, 2013 - ACS Publications
Scope and limitations in the diastereoselective preparation of 2, 6-cis or 2, 6-trans
disubstituted piperidines are described, through intramolecular reaction of chiral β …

Synthesis of 2, 6-disubstituted piperidine alkaloids from ladybird beetles Calvia 10-guttata and Calvia 14-guttata

P Kubizna, I Špánik, J Kožíšek, P Szolcsányi - Tetrahedron, 2010 - Elsevier
Optically pure (+)-calvine,(+)-2-epicalvine,(2S, 6S)-(6-pentylpiperidin-2-yl) acetic acid methyl
ester and (2R, 6S)-(6-pentylpiperidin-2-yl) acetic acid methyl ester, four piperidine alkaloids …

Domino Imino-Aldol− Aza-Michael Reaction: One-Pot Diastereo-and Enantioselective Synthesis of Piperidines

MK Ghorai, S Halder, RK Das - The Journal of Organic Chemistry, 2010 - ACS Publications
Addition of α-arylmethylidene-or α-alkylidene-β-keto ester enolate to N-activated aldimines
via the imino aldol pathway followed by intramolecular aza-Michael reaction in a domino …

[HTML][HTML] Stereoselective Allylic Alkylations of Amino Ketones and Their Application in the Synthesis of Highly Functionalized Piperidines

C Prudel, K Huwig, U Kazmaier - Chemistry (Weinheim an der …, 2020 - ncbi.nlm.nih.gov
Stereoselective Allylic Alkylations of Amino Ketones and Their Application in the Synthesis of
Highly Functionalized Piperidines - PMC Back to Top Skip to main content NIH NLM Logo …

Stereocontrolled reduction of chiral pyrrolidine and piperidine β-enamino esters: formal enantioselective synthesis of (+)-calvine

S Calvet-Vitale, C Vanucci-Bacqué… - Tetrahedron, 2005 - Elsevier
Stereocontrolled reduction of chiral pyrrolidine and piperidine β-enamino esters: formal
enantioselective synthesis of (+)-calvine - ScienceDirect Skip to main contentSkip to article …

β-Amino acids to piperidinones by Petasis methylenation and acid-induced cyclization

LV Adriaenssens, RC Hartley - The Journal of Organic Chemistry, 2007 - ACS Publications
Ester-imine derivatives of β-amino acids were methylenated with dimethyltitanocene under
microwave irradiation and the resulting enol ethers cyclized with Brönsted acid or …

Short racemic syntheses of calvine and epicalvine

P Szolcsányi, T Gracza, I Špánik - Tetrahedron Letters, 2008 - Elsevier
The intramolecular Pd (II)-catalysed carbonylation of aminoalkenitol was used as a key step
in the short racemic syntheses of the ladybird beetle alkaloids calvine and epicalvine. The …