Covering the fundamentals of heterocyclic reactivity and synthesis, this book teaches the
subject in a way that is understandable to graduate students. Recognizing the level at which …

This review presents the recent progress in the chemistry of dimethyl acetylenedicarboxylate
(DMAD). The interest in and applications of this powerful reagent with more than 135 years …

This review reports the reactivity of indolizines. The reactions section covers, in general,
electrophilic, oxidation, reduction, addition, cycloaddition, condensation, and Mannich and …

The first enantioselective [12+ 2] cycloaddition has been developed for the construction of a
chiral cycl [3.2. 2] azine core, a tricyclic moiety with a central ring-junction nitrogen atom, by …

A variety of C-2 and C-5 difunctionalized indolizines have been prepared through the
reaction of 1-ester-substituted indolizines with organometallic bases followed by a reaction …

The reaction between benzynes and imidazo [1, 2-a] pyridines (pyrimidines) to form benzo
[a] imidazo [5, 1, 2-cd] indolizines and 2, 3, 9c-triazocyclopenta [j, k] fluorenes has been …

Herein we reported the synthesis of 20 novel fluorescent 5-carbonylated 2-arylindolizines
derivatives through the reaction between organolithium intermediates with different …

A dehydrogenative Heck annelation reaction of indolizine with diaryl acetylene via dual C–H
bond cleavage was developed. Oxygen gas was employed as a clean oxidant in this …

3-Haloindolizines were synthesized via Cu (II) halide mediated halogenation of indolizines.
This C− H direct functionalization process occurred under mild conditions giving 3 …

The C–H borylation of indolizines has not previously been reported. In this communication,
we describe our preliminary efforts to apply this chemistry to this scaffold and contrast this …