In vitro and in silico studies of fluorinated 2, 3‐disubstituted thiazolidinone‐pyrazoles as potential α‐amylase inhibitors and antioxidant agents
As part of our effort to identify potent α‐amylase inhibitors, in the present study, a novel
series of fluorinated thiazolidinone‐pyrazole hybrid molecules were prepared by the …
series of fluorinated thiazolidinone‐pyrazole hybrid molecules were prepared by the …
Design, synthesis and anti-microbial activity of 1H-pyrazole carboxylates
In a SAR study, we have synthesized a few 1H-pyrazole carboxylate related microbicides
using Vilsmeier reagent. The anti-microbial screening results of 1H-pyrazole-3-carboxylate …
using Vilsmeier reagent. The anti-microbial screening results of 1H-pyrazole-3-carboxylate …
The Vilsmeier reaction of non‐aromatic compounds
G Jones, SP Stanforth - Organic Reactions, 2004 - Wiley Online Library
This chapter extends the discussion to reactions between the Vilsmeier‐Haack reagent
(subsequently referred to as the Vilsmeier reagent for brevity) and any other compounds in …
(subsequently referred to as the Vilsmeier reagent for brevity) and any other compounds in …
Product class 1: pyrazoles
B Stanovnik, J Svete - Science of Synthesis, 2002 - thieme-connect.com
Previously published information regarding this heterocyclic system can be found in
Houben±Weyl, Vol. 13/6, pp 181±522 and Vol. 22b, pp 1508±1516. Pyrazole (1, 2-diazole) …
Houben±Weyl, Vol. 13/6, pp 181±522 and Vol. 22b, pp 1508±1516. Pyrazole (1, 2-diazole) …
Cyclizations under Vilsmeier conditions
O Meth-Cohn, B Tarnowski - Advances in Heterocyclic Chemistry, 1982 - Elsevier
Publisher Summary The Vilsmeier—or Vilsmeier-Haack or Vilsmeier-Haack-Arnold—
reaction is primarily a mild method for formulating a wide variety of substrates. It has a …
reaction is primarily a mild method for formulating a wide variety of substrates. It has a …
[图书][B] Synthesis using Vilsmeier reagents
CM Marson - 2018 - taylorfrancis.com
Synthesis Using Vilsmeier Reagents presents a comprehensive account of the whole of
Vilsmeier chemistry, including the formation of over 50 functional groups and over 50 …
Vilsmeier chemistry, including the formation of over 50 functional groups and over 50 …
Molecular design of pyrazolo[3,4-d]pyridazines
VS Matiichuk, MA Potopnyk, ND Obushak - Russian Journal of Organic …, 2008 - Springer
Reactions of arenediazonium chlorides with ethyl 2-methyl-and 2-chloro-4-oxobutanoates
gave, respectively, ethyl 2-(arylhydrazono) propanoates and chloro (arylhydrazono) …
gave, respectively, ethyl 2-(arylhydrazono) propanoates and chloro (arylhydrazono) …
A concise review on the synthesis of pyrazole heterocycles
AM Dar, S Shamsuzzaman - 2015 - hero.epa.gov
Pyrazole moiety, being called as pharmacophore, plays an important role in many
biologically active compounds and therefore represents an interesting template for …
biologically active compounds and therefore represents an interesting template for …
Synthesis of Novel 1-H-Pyrazole-4-carboxylic Acid Esters by Conventional and Microwave Assisted Vilsmeier Cyclization of Hydrazones
R Sridhar, PT Perumal - Synthetic communications, 2003 - Taylor & Francis
Full article: Synthesis of Novel 1-H-Pyrazole-4-carboxylic Acid Esters by Conventional and
Microwave Assisted Vilsmeier Cyclization of Hydrazones Skip to Main Content Taylor and …
Microwave Assisted Vilsmeier Cyclization of Hydrazones Skip to Main Content Taylor and …
Synthesis and inhibitory activity of 4-alkynyl and 4-alkenylquinazolines: Identification of new scaffolds for potent EGFR tyrosine kinase inhibitors
Y Kitano, T Suzuki, E Kawahara, T Yamazaki - Bioorganic & medicinal …, 2007 - Elsevier
The present study identified several 4-alkynyl and 4-alkenylquinazolines that serve as novel
and potent EGFR tyrosine kinase inhibitors. The IC50 values of these compounds are in the …
and potent EGFR tyrosine kinase inhibitors. The IC50 values of these compounds are in the …