Berberine derivatives as inhibitors of acetylcholinesterase: A systematic review

YP Singh, H Kumar - Chemical Biology & Drug Design, 2023 - Wiley Online Library
Alzheimer's disease (AD) is a chronic age‐related neurodegenerative brain disorder
characterized by the impairment of memory accompanied by worsening of thinking ability of …

In Vitro and In Silico Evaluation of Amylase, Tyrosinase, and Pancreatic Lipase Inhibitions of Novel Benzothiazole‐Sulfonate Derivatives

A Korkmaz, E Bursal, G Kurtay - ChemistrySelect, 2023 - Wiley Online Library
This paper provides a comprehensive account of the synthesis and assessment of newly
developed aryl sulfonate derivatives based on benzothiazole as enzyme inhibitors …

Sulfonyl thioureas with a benzo[d]thiazole ring as dual acetylcholinesterase/butyrylcholinesterase and human monoamine oxidase A and B inhibitors: An in vitro and …

N Dinh Thanh, D Son Hai, V Ngoc Toan… - Archiv der …, 2024 - Wiley Online Library
A series of sulfonyl thioureas 6a–q containing a benzo [d] thiazole ring with an ester
functional group was synthesized from corresponding substituted 2‐aminobenzo [d] …

Eco‐friendly Regioselective Synthesis, Biological Evaluation of Some New 5‐acylfunctionalized 2‐(1H‐pyrazol‐1‐yl)thiazoles as Potential Antimicrobial and …

R Aggarwal, M Sharma, M Hooda, PC Sharma… - …, 2024 - Wiley Online Library
The present study describes an eco‐friendly NBS‐assisted regioselective synthesis of new 5‐
acylfunctionalized 5‐acylfunctionalized 2‐(1H‐pyrazol‐1‐yl) thiazoles by condensation of 3 …

抗阿尔茨海默病噻唑衍生物的设计策略及构效关系研究进展

史大华, 邹靖培, 张笑清, 张钊源… - 河北大学学报(自然科学版), 2024 - xbzrb.hbu.edu.cn
噻唑是一种五元含硫, 氮杂环化合物, 由于其特殊的结构和电子性质以及具有的多种生物学活性,
已成为药物化学领域中广泛运用的化学骨架之一. 在过去的几十年里, 噻唑及其衍生物在抗阿尔 …