Several naturally occurring purine and pyrimidine nucleosides contain an amide linkage as
part of the heterocyclic aglycone. Enolization of the amide and conversion to leaving groups …

Despite the impressive progress in nucleoside chemistry to date, the synthesis of nucleoside
analogues is still a challenge. Chemoenzymatic synthesis has been proven to overcome …

Deaminative modifications of purines via diazonium chemistry have long been the
cornerstone in modified nucleoside synthesis. The purpose of this review is to bring into …

Reactions of Ot-butyldimethylsilyl-protected thymidine, 2′-deoxyuridine, and 3′-
azidothymidine (AZT) with (benzotriazol-1-yloxy) tris (dimethylamino) phosphonium …

Abstract Ethyl 3-tert-butyl-4-oxo-7-X-4, 6-dihydropyrazolo [5, 1-c][1, 2, 4] triazine-8-
carboxylates (X= H, Cl, Br) were synthesized for the first time by diazotization of 7-amino-3 …

The synthesis and catalytic applications of the highly water‐soluble ligand 7‐phospha‐1, 3,
5‐triaza‐admantane butane sultonate (PTABS) has been described. The synthesized …

1, 4‐Triazolyl combretacoumarins have been prepared by linking the trimethoxyarene unit of
combretastatin A4 with coumarins, via a 1, 2, 3‐triazole. For this, 4‐azidocoumarins were …

Этил-3-трет-бутил-4-оксо-7-X-4, 6-дигидропиразоло [5, 1-c][1, 2, 4] триазин-8-
карбоксилаты (X= H, Cl, Br) впервые синтезированы диазотированием 7-амино-3-трет …

Reaction of amide bonds in t-butyldimethylsilyl-protected inosine, 2′-deoxyinosine,
guanosine, 2′-deoxyguanosine, and 2-phenylinosine with commercially available peptide …

N 6-methyladenosine (m6A) is the most abundant modification in mRNA. Studies on
proteins that introduce and bind m6A require the efficient synthesis of oligonucleotides …