As one of the most important structural units in pharmaceuticals and medicinal chemistry,
quinazolinone and its derivatives exhibit a wide range of biological and pharmacological …

This review highlights recent progress in electrochemical cascade cyclization reactions for
the synthesis of carbon rings and heterocycles, such as pyridines, quinolines …

An efficient radical cascade cyclization of unactivated alkenes toward the synthesis of a
series of ring-fused quinazolinones has been developed in moderate to excellent yields …

The dehydrogenative cross‐coupling reaction is the premier route for synthesizing important
4‐quinazolinone drugs. However, it usually requires high reaction temperature and long …

A transition-metal-free C═ C double bond cleavage reaction employing molecular iodine is
described. In the presence of K2CO3 as the base, I2-mediated C═ C bond cleavage …

A novel cascade radical addition/cyclization reaction of non-activated olefins and oxamic
acids has been proposed. Under transition metal-free conditions, 36 quinazolinone …

A simple metal-free method for the synthesis of quinazolinones from commercially available
2-nitrobenzyl alcohols and tetrahydroisoquinolines is developed. The reaction conditions …

New photochemical approaches to 2, 3-fused quinazolinones and dihydroquinazolinones
are disclosed. The intramolecular hydrocyclization proceeds in moderate to excellent yields …

We report herein an efficient and practical strategy for the preparation of 5 H-phthalazino [1,
2-b] quinazolin-8 (6 H)-one derivatives through at-BuOK-catalyzed intramolecular …

The incorporation of amide groups into biologically active molecules has been proven to be
an efficient strategy for drug design and discovery. In this study, we present a simple and …