Recent advances in the cascade reactions of enynols/diynols for the synthesis of carbo-and heterocycles

S Jiang, H Ma, R Yang, XR Song, Q Xiao - Organic Chemistry Frontiers, 2022 - pubs.rsc.org
Carbo-and heterocycles frequently serve as crucial scaffolds in drugs, natural products, fine
chemicals, and biologically and pharmaceutically active compounds. Consequently, the …

Multicomponent reactions of ethyl trifluoroacetoacetate with carbonyl and nucleophilic reagents as a promising tool for organic synthesis

SO Kushch, MV Goryaeva, YV Burgart… - Russian Chemical …, 2023 - Springer
The review is summarized and systematized the published data on the multicomponent
reactions of ethyl trifluoroacetoacetate, carbonyl compounds (aldehydes and ketones), and …

Copper-catalyzed divergent construction of naphthofurans and benzochromanes from 2-naphthols, 4-methylene-quinazolin (thi) ones, and N, N-dimethylethanolamine

M Geng, J Kuang, W Fang, X Xiao, Y Ma - Organic Chemistry Frontiers, 2024 - pubs.rsc.org
We report herein an unprecedented Cu (II)-catalyzed divergent synthesis of naphthofurans
and benzochromanes from 2-naphthols, N, N-dimethylethanolamine, and methylene-3, 4 …

Organocatalytic (Z/E)-Selective Synthesis of 3-Vinylnaphthofurans via a Formal (3 + 2) Cycloaddition

L Yu, R Xu, YY Yao, Y Lu, FY Liu… - The Journal of Organic …, 2023 - ACS Publications
A formal (3+ 2) cycloaddition of 1, 4-enediones with 2-naphthols was established under the
catalysis of trifluoromethanesulfonic acid as an organocatalyst, leading to the efficient …

Indole frameworks via transition-metal-free annulation: a current perspective

S Das - New Journal of Chemistry, 2023 - pubs.rsc.org
Indole structural motifs are ubiquitous in natural products, pharmaceuticals, agrochemicals
and functional materials. The immense importance of the indole moiety, especially in the …

Direct C–C Bond Cleavage of 1, 3-Dicarbonyl Compounds as a Single-Carbon Synthon: Synthesis of 2-Aryl-4-quinolinecarboxylates

Y Zhou, P Zhao, LS Wang, XX Yu, C Huang… - Organic …, 2021 - ACS Publications
A novel [2+ 1+ 3] cyclization reaction for the synthesis of 2-aryl-4-quinolinecarboxylates from
aryl methyl ketones, arylamines, and 1, 3-dicarbonyl compounds has been established. This …

One-Pot Synthesis of N-Fused Benzimidazo-β-carbolines through Sequential Propargylation/aza-Cycloisomerization Approach

CR Reddy, K Nair, E Srinivasu… - The Journal of Organic …, 2024 - ACS Publications
The first sequential acid-catalyzed propargylation/base-mediated aza-cycloisomerization
between indolyl-benzimidazoles and propargylic alcohols is described. This protocol …

A Domino Dearomative ipso-Annulation/Desymmetrization Approach: Stereoselective Access to Tricyclic Alkaloid Skeletons

CR Reddy, AS Prasad, U Ajaykumar - Organic Letters, 2024 - ACS Publications
Herein, we reveal an unprecedented domino annulation of N-benzyl-acrylamides with 1, 3-
dicarbonyls for the assembly of fused tricyclic alkaloid frameworks incorporating a spirocycle …

A Comprehensive Review on Benzofuran Synthesis Featuring Innovative and Catalytic Strategies

A Mushtaq, AF Zahoor, S Ahmad, MJ Saif, A ul Haq… - ACS …, 2024 - ACS Publications
Benzofurans have intrigued both pharmaceutical researchers and chemists owing to the
medicinal usage of their derivatives against copious disease-causing agents (ie, bacteria …

FeCl 3-mediated selenylative benzannulation of aryl alkynones to 3-selenyl β-naphthols

CR Reddy, MC Bhandari, AD Patil, M Aila… - Organic & Biomolecular …, 2022 - pubs.rsc.org
An efficient selenylative cyclization of aryl-alkynones with diselenides in the presence of iron
(III) chloride at room temperature to prepare 3-seleno-2-naphthols in good yields has been …