In the past two decades, transition metal-catalyzed C–H functionalization followed by
annulations with various coupling partners has received much attention in organic synthesis …

The cyclohepta [b] indole scaffold constitutes a salient structural motif in natural products as
well as in men‐made pharmaceutically active ingredients. Cyclohepta [b] indoles consist of …

Highly selective and switchable [4+ 2] annulations of 2-arylindoles with iodonium ylides
were achieved by performing solvent-controlled Rh (III)-catalyzed C–H activations. When …

A robust metal-free and environmentally friendly approach to cyclohepta [b] indole and furo
[3, 4-b] carbazole frameworks via a three-component reaction from indoles, tertiary …

Chemodivergent synthesis of indeno [1, 2-b] indoles and isoindolo [2, 1-a] indoles from the
same starting materials involving radical cross-dehydrogenative couplings have been …

An efficient acid-catalyzed three-component cascade strategy was established on the basis
of a crucial conversion of BIMs to vinylindoles to synthesize a privileged scaffold, phenyl …

The treatment of many bacterial diseases remains a significant problem due to the
increasing antibiotic resistance of their infectious agents. Among others, this is related to …

We report herein the facile synthesis of indole-fused six-, seven-, or eight-membered N, O-
heterocycles through rhodium-catalyzed C–H acetoxylation/hydrolysis/annulation. The …

Here, Selective C3-formylation of indole was achieved under mild conditions using a metal–
organic framework (MOF) catalyst. The confined reaction space within the MOF pores …

Diversity-oriented synthesis strategy for the efficient assembly of indole-fused polycyclic
scaffolds via rhodium-catalyzed NH-indole-directed C–H coupling with propargylic alcohol …