Hydrogenolysis of N-protected aminooxetanes over palladium: An efficient method for a one-step ring opening and debenzylation reaction

E Kovács, A Thurner, F Farkas, F Faigl… - Journal of Molecular …, 2011 - Elsevier
An efficient method for the palladium mediated hydrogenation of an optically active, N-
protected aminooxetane derivative has been developed. Using appropriate solvents, in a …

[PDF][PDF] Synthesis and application of new optically active compounds as catalysts and ligands in enantioselective reactions

B MátRAvöLgyi, E KOváCS, L Hegedűs… - PERIODICA …, 2015 - real.mtak.hu
New methods for efficient preparation of optically active compounds developed recently are
reported. Combination of selective organometallic, organocatalytic, phase transfer catalytic …

Novel stereoselective synthesis of 1, 2, 3-trisubstituted azetidines

F Faigl, E Kovács, G Turczel, Á Szöllősy, A Mordini… - Tetrahedron …, 2012 - Elsevier
A novel, superbase induced diastereoselective transformation of benzylamino groups
containing oxiranes has provided a series of trans-1, 2, 3-trisubstituted azetidines in good …

First total synthesis of (+)-epogymnolactam, a novel autophagy inducer

Y Okado, K Shigetomi, S Mitsuhashi… - The Journal of …, 2015 - nature.com
Abstract A novel autophagy inducer,(+)-epogymnolactam (1), was first synthesized from cis-
4-benzyloxy-2-butene-1-ol (2) in eight steps. A reliable preparation of optically pure epoxy …

Synthesis and enantioselective rearrangement of (Z)‐4‐triphenylmethoxy‐2,3‐epoxybutan‐1‐ol enantiomers

F Faigl, A Thurner, F Farkas… - Chirality: The …, 2007 - Wiley Online Library
Efficient enzyme catalyzed kinetic resolutions of a synthetically useful chiral building
block,(Z)‐4‐triphenylmethoxy‐2, 3‐epoxybutan‐1‐ol, are reported. The highest selectivities …

Solvent-dependent reactivity in porcine pancreatic lipase (PPL)-catalyzed hydrolysis

LL Shen, F Wang, HS Mun, M Suh, JH Jeong - Tetrahedron: Asymmetry, 2008 - Elsevier
The solvent-dependent enzyme reactivity of porcine pancreatic lipase (PPL)-catalyzed
hydrolysis was investigated using trans-3 and cis-(3-(benzyloxymethyl) oxiran-2-yl) methyl …

Four-membered ring systems

B Alcaide, P Almendros - Progress in Heterocyclic Chemistry, 2009 - Elsevier
Publisher Summary This chapter highlights the current state of the art in the vast area of four-
membered heterocyclic chemistry. There has been explosive growth in the research area of …

[PDF][PDF] Racém 2, 3-epoxibutanol-származékok rezolválása és enantioszelektív átrendeződési reakciói

F Ferenca, F Ferenca, K Ervina, T Angelikab - epa.niif.hu
A királis oxirán-és oxetán-származékok (epoxidok, oxaciklobutánok) gyakran használt
gyógyszer-és növényvédőszeripari intermedierek. Többek között antibiotikumok, 1, 2 vírus …

Multi-rotor internal rotations and conformational equilibria in oxiraneethanol and assignment of its vibrational spectra

HM Badawi, SA Ali - Journal of Molecular Structure, 2009 - Elsevier
The complex internal rotations and conformational equilibria in oxiraneethanol were
investigated at the DFT-B3LYP/6-311G** level of theory. Four minima were predicted in the …

Novel Methods for the Separation of Optical Isomers

F Faigl, B Mátravölgyi, A Thurner - New Methodologies and Techniques …, 2008 - Springer
Recent developments in the field of racemate resolution has been reviewed and illustrated
with examples. The excellent results achieved by the novel pH-controlled crystallization of …