Recent developments and biological activities of thiazolidinone derivatives: A review

AK Jain, A Vaidya, V Ravichandran, SK Kashaw… - Bioorganic & medicinal …, 2012 - Elsevier
Thiazolidinone is considered as a biologically important active scaffold that possesses
almost all types of biological activities. Successful introduction of ralitoline as a potent anti …

4-Thiazolidinones: the advances continue…

AC Tripathi, SJ Gupta, GN Fatima, PK Sonar… - European Journal of …, 2014 - Elsevier
The diversity in the biological response of 4-thiazolidinones has attracted the attention of
many researchers to explore this framework for its potential. It is, therefore, of prime …

Rapid, selective heavy metal removal from water by a metal–organic framework/polydopamine composite

DT Sun, L Peng, WS Reeder, SM Moosavi… - ACS central …, 2018 - ACS Publications
Drinking water contamination with heavy metals, particularly lead, is a persistent problem
worldwide with grave public health consequences. Existing purification methods often …

Therapeutic role of nitric oxide as emerging molecule

S Kumar, RK Singh, TR Bhardwaj - Biomedicine & Pharmacotherapy, 2017 - Elsevier
NO has many physiological roles; in inflammation, pain, rheumatoid arthritis, immune
system, gastroprotection, as antioxidant and reported to be a free radical scavenger …

Epihalohydrins in organic synthesis

GS Singh, K Mollet, M D'hooghe… - Chemical Reviews, 2013 - ACS Publications
Epihalohydrins [2-(halomethyl) oxiranes, 1, 2-epoxy-3-halopropanes](Figure 1) are well-
known versatile synthons and important reagents in the realm of organic synthesis …

Open source drug discovery: highly potent antimalarial compounds derived from the tres cantos arylpyrroles

AE Williamson, PM Ylioja, MN Robertson… - ACS central …, 2016 - ACS Publications
The development of new antimalarial compounds remains a pivotal part of the strategy for
malaria elimination. Recent large-scale phenotypic screens have provided a wealth of …

Antiproliferative activity and molecular docking studies of new 4-oxothiazolidin-5-ylidene acetate derivatives containing guanylhydrazone moiety

IAS Al-Janabi, SÇ Yavuz, S Köprü, M Tapera… - Journal of Molecular …, 2022 - Elsevier
A new series of 4-oxothiazolidin-5-ylidene acetates (1–16) containing guanylhydrazone
moiety were designed and synthesized by using dimethyl acetylenedicarboxylate (DMAD) …

Discovery of a selective aurora a kinase inhibitor by virtual screening

F Kilchmann, MJ Marcaida, S Kotak… - Journal of medicinal …, 2016 - ACS Publications
Here we report the discovery of a selective inhibitor of Aurora A, a key regulator of cell
division and potential anticancer target. We used the atom category extended ligand overlap …

An efficient One-pot three-component synthesis, Molecular docking, ADME and DFT predictions of new series Thiazolidin-4-one derivatives bearing a Sulfonamide …

SA Hassan, DM Aziz - Egyptian Journal of Chemistry, 2022 - journals.ekb.eg
As part of our endeavor to synthesize a new series of biologically effective heterocyclic
hybrids, we present various methods for one-pot three-component synthesis. The thiazolidin …

Antiproliferative and tumor inhibitory studies of 2, 3 disubstituted 4-thiazolidinone derivatives

KSS Kumar, A Hanumappa, M Vetrivel, M Hegde… - Bioorganic & medicinal …, 2015 - Elsevier
Thiazolidinone derivatives were synthesized using T3P®-DMSO media as a
cyclodehydrating agent. All the molecules were tested for their cytotoxicity against leukemic …