Synthetic approaches, functionalization and therapeutic potential of quinazoline and quinazolinone skeletons: The advances continue

I Khan, A Ibrar, W Ahmed, A Saeed - European journal of medicinal …, 2015 - Elsevier
The presence of N-heterocycles as an essential structural motif in a variety of biologically
active substances has stimulated the development of new strategies and technologies for …

Recent advances in the synthesis of Quinazoline analogues as Anti-TB agents

A Dutta, D Sarma - Tuberculosis, 2020 - Elsevier
Quinazoline analogues are one of the important nitrogen containing heterocycles that have
significant bioactivity as well as found in a plethora of natural products. Tuberculosis is one …

Synthesis and photophysical studies of a series of quinazoline chromophores

S Achelle, J Rodrı́guez-López… - The Journal of Organic …, 2014 - ACS Publications
The synthesis of a series of push–pull arylvinyl (styryl), aryl, and arylethynyl quinazoline
derivatives by means of different straightforward protocols is reported. The photophysical …

Influence of the Base on Pd@MIL‐101‐NH2(Cr) as Catalyst for the Suzuki–Miyaura Cross‐Coupling Reaction

F Carson, V Pascanu, A Bermejo Gómez… - … A European Journal, 2015 - Wiley Online Library
The chemical stability of metal–organic frameworks (MOFs) is a major factor preventing their
use in industrial processes. Herein, it is shown that judicious choice of the base for the …

Effect of protonation on the photophysical properties of 4-substituted and 4, 7-disubstituted quinazoline push-pull chromophores

R Plaza-Pedroche, D Georgiou, M Fakis, A Fihey… - Dyes and …, 2021 - Elsevier
White-light emission from single molecular systems has attracted a great deal of attention
due to their advantages over multicomponent emitters. Azaheterocyclic push-pull derivatives …

[HTML][HTML] Pd-, Cu-, and Ni-Catalyzed Reactions: A Comprehensive Review of the Efficient Approaches towards the Synthesis of Antibacterial Molecules

A Zia, S Khalid, N Rasool, N Mohsin, M Imran, SI Toma… - Pharmaceuticals, 2024 - mdpi.com
A strong synthetic tool for many naturally occurring chemicals, polymers, and
pharmaceutical substances is transition metal-catalyzed synthesis. A serious concern to …

[PDF][PDF] Review on synthesis schemes of first line drugs of antitubercular drugs

V Sahu, V Kushwaha, V Sahu, S Shukla… - Indian Journal of Science …, 2022 - ijsronline.org
Review Article Page 1 Sahu V et al., Ind. J. Sci. Res. 2022, 2(2), 53-59 Indian Journal of
Science and Research. Vol.2 Issue-2 - 53 - [ISSN 2583-2913] Review Article *Corresponding …

Kumada cross coupling reaction for the synthesis of quinazoline derivatives, evaluation of their antibacterial activity and docking studies

AR Ankireddy, R Syed, R Gundla, KL Manasa… - Russian Journal of …, 2019 - Springer
A series of C7-substituted-2-morpholino-N-(pyridin-2-ylmethyl) quinazolin-4-amine
derivatives 3a–3t were synthesized by using Nickel catalyzed Kumada cross coupling …

Suzuki–Miyaura coupling of quinazolines containing an unprotected NH2 group: Synthesis and biological testing of quinazoline derivatives

Y Pulipati, V Gurram, SV Laxmi… - Synthetic …, 2017 - Taylor & Francis
ABSTRACT A robust approach to 4-amino quinazoline bi-aryl compounds was developed
through Suzuki–Miyaura coupling reaction of quinazoline containing an unprotected NH2 …

[PDF][PDF] Design, synthesis, antitumor and antimicrobial activity of novel 6, 7-dimethoxyquinazoline derivatives

AE Kassab, EM Gedawy, Z Mahmoud… - …, 2016 - triggered.stanford.clockss.org
Novel 4-substituted-6, 7-dimethoxyquinazolines 3, 4a and 4b were synthesized via reacting
the corresponding 4-chloro derivative 2 with 2-(4-aminopiperazin-1-yl) ethanol …