Biologically active azolo-1, 2, 4-triazines and azolopyrimidines

VL Rusinov, VN Charushin, ON Chupakhin - Russian Chemical Bulletin, 2018 - Springer
The review presents current data on the methods of synthesis and biological activity of
purine-isosteric azolo-annulated 1, 2, 4-triazines and pyrimidines with a bridgehead …

Modern Trends of Organic Chemistry in Russian Universities

AI Konovalov, IS Antipin, VA Burilov… - Russian Journal of …, 2018 - Springer
This review is devoted to the scientific achievements of the departments of organic chemistry
in higher schools of Russia within the past decade.

Design, synthesis, molecular modelling, ADME prediction and anti-hyperglycemic evaluation of new pyrazole-triazolopyrimidine hybrids as potent α-glucosidase …

V Pogaku, K Gangarapu, S Basavoju, KK Tatapudi… - Bioorganic …, 2019 - Elsevier
The aim of the present study is to design and synthesis of new pyrazole-triazolopyrimidine
hybrids as potent α-glucosidase inhibitors. The target compounds 4a-n were synthesized by …

Organic chemistry. History and mutual relations of universities of Russia

IS Antipin, MA Kazymova, MA Kuznetsov… - Russian Journal of …, 2017 - Springer
The review describes the history of development of organic chemistry in higher schools of
Russia over a period of 170 years, since the emergence of organic chemistry in our country …

6‐Nitroazolo[1,5‐a]pyrimidin‐7(4H)‐ones as Antidiabetic Agents

AA Spasov, DA Babkov, VA Sysoeva… - Archiv der …, 2017 - Wiley Online Library
Prevention of the formation of advanced glycation end‐products (AGEs) is a reliable
approach to achieve control over hyperglycemia and the associated pathogenesis of …

Pyrazolotriazines: Biological activities, synthetic strategies and recent developments

SR Alizadeh, MA Ebrahimzadeh - European Journal of Medicinal Chemistry, 2021 - Elsevier
Highlights•Pyrazolotriazine is as an attractive scaffold for drug design development.•
Biological activity (in vitro and in vivo) of these derivatives are reviewed.•The SAR studies …

Fused azoloazines with antidiabetic activity

VL Rusinov, IM Sapozhnikova, AA Spasov… - Russian Chemical …, 2022 - Springer
The purpose of this review is to summarize drugs containing an azoloazine moiety and
exhibiting antidiabetic activity. The review includes azoloazines active against dipeptidyl …

Methods of synthesis for the azolo [1, 2, 4] triazines

EK Voinkov, RA Drokin, EN Ulomsky… - Chemistry of …, 2020 - Springer
The review summarizes and analyzes data from modern information sources on the
methods of synthesis of azolo [X, Yc][1, 2, 4] triazines. Approaches to the construction of the …

[PDF][PDF] Современные тенденции органической химии в университетах России

АИ Коновалов, ИС Антипин, ВА Бурилов… - Журнал …, 2018 - researchgate.net
5. Кафедра органической химии Московского государственного университета им. МВ
Ломоносова. 6. Кафедра химии Российского национального исследовательского …

Nitrothiadiazolo [3, 2-a] pyrimidines as promising antiglycating agents

K Savateev, V Fedotov, I Butorin, O Eltsov… - European journal of …, 2020 - Elsevier
Managing the advanced glycation end-products (AGEs) concentration is a reliable approach
to achieve control over the pathogenesis of diabetic vascular complications. Inhibition of …