Imidazole and thiadiazole derivatives display an extensive application in pharmaceutical
chemistry, and they have been investigated as bioactive molecules for medicinal chemistry …

Despite significant developments in therapeutic strategies, Diabetes Mellitus remains an
increasing concern, leading to various complications, eg, cataracts, neuropathy, retinopathy …

In this research, rational design, synthesis, carbonic anhydrases (CAs) inhibitory effects, and
cytotoxicities of the 4-(3-(2-arylidenehydrazine-1-carbonyl)-5-(thiophen-2-yl)-1 H-pyrazole-1 …

The purpose of this study was to synthesize imidazo [2, 1‐b] thiazole derivatives,
characterize them with spectroscopical techniques and investigate for cytotoxic and …

Hepatitis C Virus (HCV), affecting millions of people worldwide, is the leading cause of liver
disorder, cirrhosis, and hepatocellular carcinoma. HCV is genetically diverse having eight …

In this study, new bis‐1, 2, 3‐triazole derivatives, N, N′‐(1, 3‐phenylene) bis (2‐(4‐R‐1H‐
1, 2, 3‐triazol‐1‐yl) acetamide), were synthesized by copper‐catalyzed azide‐alkyne …

The enantioselective copper-catalyzed borylacylation of aryl olefins with acyl chlorides and
bis-(pinacolato) diboron is reported. This three-component reaction involves an …

A rhodium-catalyzed tandem arylation/cyclization reaction of 3-(ortho-boronated aryl)
conjugated enones with unactivated alkynes is reported. By using a rhodium (I)/chiral-diene …

Over the past decades, designing of privileged structures has emerged as a useful approach
to the discovery and optimisation of novel biologically active molecules, and many have …

Here, we prepared several dipeptides containing 2‐aminoindane‐2‐carboxylic acid (Aic)
and carried out further synthetic transformations. Synthesis and purification of modified …